日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Structural Investigation of the Interaction between a GC-376-Based Peptidomimetic PROTAC and Its Precursor with the Viral Main Protease of Coxsackievirus B3

对基于 GC-376 的肽模拟 PROTAC 及其前体与柯萨奇病毒 B3 病毒主蛋白酶相互作用的结构研究

De Santis, Alessia; Grifagni, Deborah; Orsetti, Andrea; Lenci, Elena; Rosato, Antonio; D'Onofrio, Mariapina; Trabocchi, Andrea; Ciofi-Baffoni, Simone; Cantini, Francesca; Calderone, Vito

Targeting z-Crystallin by aspirin restores the sensitivity to cisplatin in resistant A2780 ovarian cancer cells

阿司匹林靶向 z-Crystallin 可恢复耐药卵巢癌细胞 A2780 对顺铂的敏感性

Matteo Lulli, Andrea Trabocchi, Giandomenico Roviello, Martina Catalano, Laura Papucci, Astrid Parenti, Alice Molli, Cristina Napoli, Ida Landini, Nicola Schiavone, Andrea Lapucci

Diversifying DNA-Tagged Amines by Isocyanide Multicomponent Reactions for DNA-Encoded Library Synthesis

利用异氰化物多组分反应对DNA标记胺进行多样化修饰,用于DNA编码文库合成

Willems, Suzanne; Detta, Elena; Baldini, Lorenzo; Tietz, Deniz; Trabocchi, Andrea; Brunschweiger, Andreas

Development of a GC-376 Based Peptidomimetic PROTAC as a Degrader of 3-Chymotrypsin-like Protease of SARS-CoV-2

开发基于GC-376的肽模拟PROTAC作为SARS-CoV-2 3-胰凝乳蛋白酶样蛋白酶的降解剂

Grifagni, Deborah; Lenci, Elena; De Santis, Alessia; Orsetti, Andrea; Barracchia, Carlo Giorgio; Tedesco, Filomena; Bellini Puglielli, Raffaele; Lucarelli, Francesca; Lauriola, Angela; Assfalg, Michael; Cantini, Francesca; Calderone, Vito; Guardavaccaro, Daniele; Trabocchi, Andrea; D'Onofrio, Mariapina; Ciofi-Baffoni, Simone

Oxime Linked Doxorubicin Glycoconjugates Improve the Specific Targeting of Glioblastoma in High-Grade Glioma Therapy

肟基连接的阿霉素糖缀合物可提高高级别胶质瘤治疗中对胶质母细胞瘤的特异性靶向性

Iorio, Anna Lisa; Lenci, Elena; Marzano, Chiara; Bucaletti, Elisabetta; Tirinnanzi, Bianca; Casati, Giacomo; Giunti, Laura; Dallari, Caterina; Credi, Caterina; Sardi, Iacopo; Trabocchi, Andrea

DIPG-74. TARGETING TRANSCRIPTIONAL DYSREGULATION IN DMG THROUGH CDK9 AND HDAC INHIBITOR COMBINATION THERAPY

DIPG-74. 通过 CDK9 和 HDAC 抑制剂联合疗法靶向 DMG 中的转录失调

Stone, Christopher R; Harris, Dwight D; Broadwin, Mark; Kanuparthy, Meghamsh; Nho, Ju-Woo; Yalamanchili, Keertana; Hamze, Jad; Abid, M Ruhul; Sellke, Frank W; Koliavas, Stella; Contreras-Zárate, Maria J; Jaramillo-Gomez, Jenny A; Fox, Morgan; Nguyen, Alicia; Cittelly, Diana M; Kandigian, Savannah E; Chande, Sampada; Dolezal, Darin; Tang, Tang; Wang, Dejiang; Arnal-Estapé, Anna; Cheok, Stephanie K; McGuone, Declan; Liu, Yang; Goldberg, Sarah B; Blondin, Nicholas A; Chiang, Veronica L; Nguyen, Don X; BIARD, adam; LE Ludivine, DRET; Marie, DUTREIX; Alexandre, CARPENTIER; Manon, LANCIEN; Alexandre, PELLISSIER; Marie-Anne, Debily; David, CASTEL; Jacques, GRILL; Kevin, BECCARIA; Murdaugh, Rebecca L; Shekar, Meghan; Eberl, Brittany R; Tremblay, Jack R; Richard, Rosemary U; Nguyen, Linh; Omer, Bilal; Anastas, Jamie N; Iorio, Anna Lisa; Lenci, Elena; Marzano, Chiara; Tirinnanzi, Bianca; Giunti, Laura; Fonte, Carla; Guidi, Milena; Tellini, Marco; Castelli, Barbara; Nicola, Marco Di; Trabocchi, Andrea; Sardi, Iacopo; Murdaugh, Rebecca L; Eberl, Brittany R; Richard, Rosemary U; Tremblay, Jack R; Dei-Ampeh, Alfred; Olson, Calla M; Anastas, Jamie N; Eberl, Brittany R; Murdaugh, Rebecca L; Nnyagu, Adanze N; Richard, Rosemary U; Deneen, Benjamin; Yu, Kwanha; Anastas, Jamie N

Multilayered Bioorthogonal SERS Nanoprobes Selectively Aggregating in Human Fluids: A Smart Optical Assay for β-Amyloid Peptide Quantification

多层生物正交SERS纳米探针选择性地聚集于人体体液中:一种用于β-淀粉样蛋白肽定量分析的智能光学检测方法

Dallari, Caterina; Lenci, Elena; Trabocchi, Andrea; Bessi, Valentina; Bagnoli, Silvia; Nacmias, Benedetta; Credi, Caterina; Pavone, Francesco Saverio

Identification of a short ACE2-derived stapled peptide targeting the SARS-CoV-2 spike protein

鉴定针对 SARS-CoV-2 刺突蛋白的 ACE2 衍生短肽

Lorenzo Calugi, Giulia Sautariello, Elena Lenci, Mauro Leucio Mattei, Crescenzo Coppa, Nicoletta Cini, Alessandro Contini, Andrea Trabocchi

Molecular View on the i RGD Peptide Binding Mechanism: Implications for Integrin Activity and Selectivity Profiles

RGD 肽结合机制的分子视角:对整合素活性和选择性特征的影响

Vincenzo Maria D'Amore, Greta Donati, Elena Lenci, Beatrice Stefanie Ludwig, Susanne Kossatz, Monica Baiula, Andrea Trabocchi, Horst Kessler, Francesco Saverio Di Leva, Luciana Marinelli

Design and Synthesis of Novel Raman Reporters for Bioorthogonal SERS Nanoprobes Engineering

用于生物正交SERS纳米探针工程的新型拉曼报告分子的设计与合成

Dallari, Caterina; Innocenti, Riccardo; Lenci, Elena; Trabocchi, Andrea; Pavone, Francesco Saverio; Credi, Caterina