日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pyruvate dehydrogenase kinase regulates vascular inflammation in atherosclerosis and increases cardiovascular risk

丙酮酸脱氢酶激酶调节动脉粥样硬化中的血管炎症并增加心血管风险

Forteza, Maria J; Berg, Martin; Edsfeldt, Andreas; Sun, Jangming; Baumgartner, Roland; Kareinen, Ilona; Casagrande, Felipe Beccaria; Hedin, Ulf; Zhang, Song; Vuckovic, Ivan; Dzeja, Petras P; Polyzos, Konstantinos A; Gisterå, Anton; Trauelsen, Mette; Schwartz, Thue W; Dib, Lea; Herrmann, Joerg; Monaco, Claudia; Matic, Ljubica; Gonçalves, Isabel; Ketelhuth, Daniel F J

Free fatty acid receptor 1 stimulates cAMP production and gut hormone secretion through Gq-mediated activation of adenylate cyclase 2.

游离脂肪酸受体 1 通过 Gq 介导的腺苷酸环化酶 2 的激活来刺激 cAMP 的产生和肠道激素的分泌

Petersen Jacob Emil, Pedersen Maria Hauge, Dmytriyeva Oksana, Nellemose Emilie, Arora Tulika, Engelstoft Maja Storm, Asher Wesley B, Javitch Jonathan A, Schwartz Thue W, Trauelsen Mette

G-Protein-Coupled Receptor 91-Dependent Signalling Does Not Influence Vascular Inflammation and Atherosclerosis in Hyperlipidaemic Mice

G蛋白偶联受体91依赖性信号传导不影响高脂血症小鼠的血管炎症和动脉粥样硬化

Griepke, Silke; Trauelsen, Mette; Nilsson, Michelle D; Hansen, Jakob; Steffensen, Lasse B; Schwartz, Thue W; Ketelhuth, Daniel F J

Lactate receptor GPR81 drives breast cancer growth and invasiveness through regulation of ECM properties and Notch ligand DLL4

乳酸受体 GPR81 通过调节 ECM 特性和 Notch 配体 DLL4 来驱动乳腺癌的生长和侵袭性

Kathrine Lundø, Oksana Dmytriyeva, Louise Spøhr, Eliana Goncalves-Alves, Jiayi Yao, Laia P Blasco, Mette Trauelsen, Muthulakshmi Ponniah, Marc Severin, Albin Sandelin, Marie Kveiborg, Thue W Schwartz, Stine F Pedersen

Activation of succinate receptor 1 boosts human mast cell reactivity and allergic bronchoconstriction

琥珀酸受体1的激活可增强人类肥大细胞反应性和过敏性支气管收缩

Tang, Xiao; Rönnberg, Elin; Säfholm, Jesper; Thulasingam, Madhuranayaki; Trauelsen, Mette; Schwartz, Thue W; Wheelock, Craig E; Dahlén, Sven-Erik; Nilsson, Gunnar; Haeggström, Jesper Z

Extracellular succinate hyperpolarizes M2 macrophages through SUCNR1/GPR91-mediated Gq signaling

细胞外琥珀酸通过 SUCNR1/GPR91 介导的 Gq 信号使 M2 巨噬细胞超极化

Mette Trauelsen, Thomas K Hiron, Da Lin, Jacob E Petersen, Billy Breton, Anna Sofie Husted, Siv A Hjorth, Asuka Inoue, Thomas M Frimurer, Michel Bouvier, Chris A O'Callaghan, Thue W Schwartz

Structure-Activity Investigations and Optimisations of Non-metabolite Agonists for the Succinate Receptor 1

琥珀酸受体1非代谢激动剂的结构-活性研究与优化

Rexen Ulven, Elisabeth; Trauelsen, Mette; Brvar, Matjaz; Lückmann, Michael; Bielefeldt, Line Ø; Jensen, Lisa K I; Schwartz, Thue W; Frimurer, Thomas M

Receptor structure-based discovery of non-metabolite agonists for the succinate receptor GPR91

基于受体结构的琥珀酸受体GPR91非代谢物激动剂的发现

Trauelsen, Mette; Rexen Ulven, Elisabeth; Hjorth, Siv A; Brvar, Matjaz; Monaco, Claudia; Frimurer, Thomas M; Schwartz, Thue W