日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Molecular Dynamics-Guided Design and Chemoproteomic Profiling of Covalent Kinase Activity Probes

分子动力学引导的共价激酶活性探针设计及化学蛋白质组学分析

Chakraborty, Pratyasha; Carlos, Anthony; Thomas, Trayder; Ghaby, Kyle; Fathi, Shaghayegh; Sharma, Mukta; Nguyen, Ngoc Kim; Farmwald, Mason; Blachowicz, Lydia; Yu, Shaopeng; Pillai, Kavya Smitha; Roux, Benoît; Moellering, Raymond

Diversity of Long-Lived Intermediates along the Binding Pathway of Imatinib to Abl Kinase Revealed by MD Simulations

分子动力学模拟揭示伊马替尼与Abl激酶结合途径中长寿命中间体的多样性

Paul, Fabian; Thomas, Trayder; Roux, Benoît

Conformational Changes in Tyrosine 11 of Neurotensin Are Required to Activate the Neurotensin Receptor 1

神经降压素酪氨酸 11 的构象变化是激活神经降压素受体 1 所必需的

Fabian Bumbak, Trayder Thomas, Billy J Noonan-Williams, Tasneem M Vaid, Fei Yan, Alice R Whitehead, Shoni Bruell, Martina Kocan, Xuan Tan, Margaret A Johnson, Ross A D Bathgate, David K Chalmers, Paul R Gooley, Daniel J Scott

Role of the Second Extracellular Loop of the Adenosine A1 Receptor on Allosteric Modulator Binding, Signaling, and Cooperativity

腺苷 A1 受体第二胞外环对变构调节剂结合、信号传导和协同作用的作用

Anh T N Nguyen, Elizabeth A Vecchio, Trayder Thomas, Toan D Nguyen, Luigi Aurelio, Peter J Scammells, Paul J White, Patrick M Sexton, Karen J Gregory, Lauren T May, Arthur Christopoulos