日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Orthosteric STING inhibition elucidates molecular correction of SAVI STING.

正构 STING 抑制阐明了 SAVI STING 的分子矫正

Xie Tao, Ruzanov Max, Critton David, Merselis Leidy, Naglich Joseph, Sack John S, Zhang Ping, Xie Chunshan, Tredup Jeffrey, Stine Laurel B, Messier Cameron, Hope David L, Caceres-Cortes Janet, Mueller Luciano, Dyckman Alaric J, Newitt John A, Choudhury Asmita, Wilson Stephen C

Improving the diffraction quality of heat-shock protein 47 crystals

提高热休克蛋白47晶体的衍射质量

Kish, Kevin; Cobell, Stephen; Szapiel, Nicolas; Yan, Chunhong; Newitt, John A; Tredup, Jeffrey; Rodrigo, Iyoncy; Tomasco, Elizabeth; Gao, Mian; Marsilio, Frank; Haugner, John; Lipovšek, Dasa; Deng, Bi; Bousquet, Patrick; Zhang, Yihong; Schmidt, Holly; Sheriff, Steven

Structure-Property Basis for Solving Transporter-Mediated Efflux and Pan-Genotypic Inhibition in HCV NS5B Inhibitors

解决HCV NS5B抑制剂中转运蛋白介导的外排和泛基因型抑制的结构-性质基础

Yeung, Kap-Sun; Beno, Brett R; Mosure, Kathy; Zhu, Juliang; Grant-Young, Katherine A; Parcella, Kyle; Anjanappa, Prakash; Bora, Rajesh Onkardas; Selvakumar, Kumaravel; Wang, Ying-Kai; Fang, Hua; Krause, Rudolph; Rigat, Karen; Liu, Mengping; Lemm, Julie; Sheriff, Steven; Witmer, Mark; Tredup, Jeffrey; Jardel, Adam; Kish, Kevin; Parker, Dawn; Haskell, Roy; Santone, Kenneth; Meanwell, Nicholas A; Soars, Matthew G; Roberts, Susan B; Kadow, John F

Potent Inhibitors of Hepatitis C Virus NS3 Protease: Employment of a Difluoromethyl Group as a Hydrogen-Bond Donor

丙型肝炎病毒NS3蛋白酶的强效抑制剂:利用二氟甲基作为氢键供体

Zheng, Barbara; D'Andrea, Stanley V; Sun, Li-Qiang; Wang, Alan Xiangdong; Chen, Yan; Hrnciar, Peter; Friborg, Jacques; Falk, Paul; Hernandez, Dennis; Yu, Fei; Sheaffer, Amy K; Knipe, Jay O; Mosure, Kathy; Rajamani, Ramkumar; Good, Andrew C; Kish, Kevin; Tredup, Jeffrey; Klei, Herbert E; Paruchuri, Manjula; Ng, Alicia; Gao, Qi; Rampulla, Richard A; Mathur, Arvind; Meanwell, Nicholas A; McPhee, Fiona; Scola, Paul M

The discovery of a pan-genotypic, primer grip inhibitor of HCV NS5B polymerase

发现一种泛基因型HCV NS5B聚合酶引物结合抑制剂

Eastman, Kyle J; Parcella, Kyle; Yeung, Kap-Sun; Grant-Young, Katharine A; Zhu, Juliang; Wang, Tao; Zhang, Zhongxing; Yin, Zhiwei; Beno, Brett R; Sheriff, Steven; Kish, Kevin; Tredup, Jeffrey; Jardel, Adam G; Halan, Vivek; Ghosh, Kaushik; Parker, Dawn; Mosure, Kathy; Fang, Hua; Wang, Ying-Kai; Lemm, Julie; Zhuo, Xiaoliang; Hanumegowda, Umesh; Rigat, Karen; Donoso, Maria; Tuttle, Maria; Zvyaga, Tatyana; Haarhoff, Zuzana; Meanwell, Nicholas A; Soars, Matthew G; Roberts, Susan B; Kadow, John F