日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Flupirtine Benzyl Carbamate Improves Neurocognitive Deficits and Molecular Pathology in the Cln6(nclf) Mouse.

氟吡汀苄基氨基甲酸酯可改善 Cln6(nclf) 小鼠的神经认知缺陷和分子病理。

Chaoul Victoria, Shmoury Omar, Alam Ramy, Saab Sara, Makoukji Joelle, Aridi Lynn Al, Makhoul Nadine J, Soueid Jihane, V Carmona Angelica, Simeon Princess, Trippier Paul C, Boustany Rose-Mary

Discovery of a pyridine-piperazine-based small molecule that enhances the activity of peptidase neurolysin

发现一种基于吡啶-哌嗪的小分子,可增强肽酶神经溶素的活性

ElSayed ElZorkany, Heba; Kandil, Haya; Jayaraman, Srinidhi; Aly, Asmaa; Esfahani, Shiva Hadi; Patel, Dhavalkumar; Dannecker, Dennis; Maciag, Monika; Paul, Alyssa; Lowran, Kaitlin; Kumari, Shikha; Bose, Samik; Ostrov, David A; Wu, Colin G; Dickson, Alex; Abbruscato, Thomas J; Trippier, Paul C; Orlando, Benjamin J; Karamyan, Vardan T

Announcing the 2024 ACS Division of Medicinal Chemistry Award Recipients: Celebrating Excellence in Medicinal Chemistry

公布2024年美国化学会药物化学分会奖项获得者:表彰药物化学领域的卓越成就

Türtscher, Selina; Grabner, Michael; Berger, Torsten W; Ferrins, Lori; Trippier, Paul C

Protocol for screening of small molecules in a CLN3 disease patient-specific iPSC-derived neuronal progenitor cell model.

CLN3 疾病患者特异性 iPSC 衍生神经元祖细胞模型中小分子筛选方案。

Venkatesan Ramu, Trippier Paul C

Discovery of an Aldo-Keto reductase 1C3 (AKR1C3) degrader

发现醛酮还原酶 1C3 (AKR1C3) 降解剂

Angelica V Carmona #, Shirisha Jonnalagadda #, Alfie M Case, Krishnaiah Maddeboina, Sravan K Jonnalagadda, Louise F Dow, Ling Duan, Trevor M Penning, Paul C Trippier

Synthesis and biological characterization of a 17β hydroxysteroid dehydrogenase type 10 (17β-HSD10) inhibitor

17β 羟基类固醇脱氢酶 10 型 (17β-HSD10) 抑制剂的合成及生物学表征

Louise F Dow, Rasangi Pathirage, Helen E Erickson, Edrees Amani, Donald R Ronning, Paul C Trippier

Coumarin-Based Aldo-Keto Reductase Family 1C (AKR1C) 2 and 3 Inhibitors

香豆素类醛酮还原酶家族 1C (AKR1C) 2 和 3 抑制剂

Jonnalagadda, Sravan K; Duan, Ling; Dow, Louise F; Boligala, Geetha P; Kosmacek, Elizabeth; McCoy, Kristyn; Oberley-Deegan, Rebecca; Chhonker, Yashpal Singh; Murry, Darryl J; Reynolds, C Patrick; Maurer, Barry J; Penning, Trevor M; Trippier, Paul C

Discovery of the Next Generation of Non-peptidomimetic Neurolysin Activators with High Blood-Brain Barrier Permeability: a Pharmacokinetics Study in Healthy and Stroke Animals

发现具有高血脑屏障通透性的新一代非肽类神经溶素激活剂:健康动物和中风动物的药代动力学研究

Zhang, Yong; Sharma, Sejal; Jonnalagadda, Shirisha; Kumari, Shikha; Queen, Aarfa; Esfahani, Shiva Hadi; Archie, Sabrina Rahman; Nozohouri, Saeideh; Patel, Dhavalkumar; Trippier, Paul C; Karamyan, Vardan T; Abbruscato, Thomas J

Excellence in Medicinal Chemistry: Celebrating ACS Medicinal Chemistry Division (MEDI) Awards. A Call for Nominations

表彰药物化学领域的卓越成就:庆祝美国化学会药物化学分会(MEDI)奖项。现诚邀提名。

Blanco, Maria-Jesus; Bryant-Friedrich, Amanda; Georg, Gunda; Ali, Amjad; Ornstein, Paul L; Ferrins, Lori; Trippier, Paul C

The evolution of small molecule enzyme activators

小分子酶激活剂的演变

Dow, Louise F; Case, Alfie M; Paustian, Megan P; Pinkerton, Braeden R; Simeon, Princess; Trippier, Paul C