日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of Potential Pteridin Reductase-1 Inhibitors for the Treatment of Leishmaniasis: A Bioinformatics Approach

利用生物信息学方法鉴定治疗利什曼病的潜在蝶呤还原酶-1抑制剂

Júnior, Paulo R da S R; Lima, Lúcio R de; Silva, Luciane B; Ramos, Ryan S; Sanches, Vitor H da S; Kimani, Njogu M; Trossini, Gustavo H G; Campos, Joaquín M; Lobato, Cleison C; Santos, Cleydson B R

Fragment Screening Reveals Novel Scaffolds against Sirtuin-2-Related Protein 1 from Trypanosoma brucei

片段筛选揭示了针对布氏锥虫Sirtuin-2相关蛋白1的新型支架

Gomes, Renan A; D Polêto, Marcelo; Verli, Hugo; Almeida, Vitor M; Marana, Sandro R; Bender, Andreas; Godoi, Bruna F; Rodrigues, Vinícius T L; da S Emery, Flavio; Trossini, Gustavo H G

Screening for Antileukemia Agents in FMS-like Tyrosine Kinase 3 (FLT3)-Mutated Acute Myeloid Leukemia Cells

在FMS样酪氨酸激酶3(FLT3)突变的急性髓系白血病细胞中筛选抗白血病药物

de Miranda, Livia Bassani Lins; Ferraz, Wítor Ribeiro; Lima, Keli; Carlos, Jorge Antonio Elias Godoy; Gatti, Fernando Moura; Alves, Rodrigo Heleno; Trossini, Gustavo Henrique Goulart; Machado-Neto, João Agostinho

SETDB1: an emerging target for anticancer drug development

SETDB1:抗癌药物研发的新兴靶点

Trossini, Gustavo Henrique Goulart; Hassanie, Haifa; Penteado, André Berndt; El-Hajje, Marissa

SETDB1 as a cancer target: challenges and perspectives in drug design

SETDB1作为癌症靶点:药物设计中的挑战与展望

Hassanie, Haifa; Penteado, André Berndt; de Almeida, Larissa Costa; Calil, Raisa Ludmila; da Silva Emery, Flávio; Costa-Lotufo, Leticia Veras; Trossini, Gustavo Henrique Goulart

Convergent QSAR Models for the Prediction of Cruzain Inhibitors

用于预测克鲁赞抑制剂的收敛性QSAR模型

Gonçalves, Rafael Bello; Ferraz, Witor Ribeiro; Calil, Raisa Ludmila; Scotti, Marcus Tullius; Trossini, Gustavo Henrique Goulart

Trypanosoma cruzi Sirtuin 2 as a Relevant Druggable Target: New Inhibitors Developed by Computer-Aided Drug Design

克氏锥虫 Sirtuin 2 作为相关可用药靶点:通过计算机辅助药物设计开发的新型抑制剂

Glaucio Monteiro Ferreira, Thales Kronenberger, Vinicius Gonçalves Maltarollo, Antti Poso, Fernando de Moura Gatti, Vitor Medeiros Almeida, Sandro Roberto Marana, Carla Duque Lopes, Daiane Yukie Tezuka, Sérgio de Albuquerque, Flavio da Silva Emery, Gustavo Henrique Goulart Trossini

Aporphine and isoquinoline derivatives block glioblastoma cell stemness and enhance temozolomide cytotoxicity

阿朴啡和异喹啉衍生物阻断胶质母细胞瘤细胞干细胞并增强替莫唑胺的细胞毒性

Dorival Mendes Rodrigues-Junior, Cristiano Raminelli, Haifa Hassanie, Gustavo Henrique Goulart Trossini, Givago Prado Perecim, Laia Caja, Aristidis Moustakas #, André Luiz Vettore #

Antibodies Against the Plasmodium vivax Apical Membrane Antigen 1 From the Belem Strain Share Common Epitopes Among Other Worldwide Variants

来自贝伦株的针对间日疟原虫顶端膜抗原1的抗体与其他全球变种共享共同表位

França, Ana Caroline Barbosa; Françoso, Kátia Sanches; Marques, Rodolfo Ferreira; Trossini, Gustavo H G; Gomes, Renan A; Póvoa, Marinete M; Cunha, Maristela G; Silveira, Eduardo L V; Soares, Irene S

Insights on 3D Structures of Potential Drug-targeting Proteins of SARS-CoV-2: Application of Cavity Search and Molecular Docking

利用空腔搜索和分子对接技术解析SARS-CoV-2潜在药物靶向蛋白的三维结构

Fernandes, Mariana S; da Silva, Francielly S; Freitas, Ana Carolina S G; de Melo, Eduardo B; Trossini, Gustavo H G; Paula, Fávero R