日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Impact of protein and small molecule interactions on kinase conformations

蛋白质和小分子相互作用对激酶构象的影响

Valentina Kugler #, Selina Schwaighofer #, Andreas Feichtner, Florian Enzler, Jakob Fleischmann, Sophie Strich, Sarah Schwarz, Rebecca Wilson, Philipp Tschaikner, Jakob Troppmair, Veronika Sexl, Pascal Meier, Teresa Kaserer, Eduard Stefan

Tracking and blocking interdependencies of cellular BRAF-MEK oncokinase activities

追踪和阻断细胞BRAF-MEK癌激酶活性的相互依赖性

Fleischmann, Jakob; Schwaighofer, Selina; De Falco, Louis; Enzler, Florian; Feichtner, Andreas; Kugler, Valentina; Tschaikner, Philipp; Huber, Roland G; Stefan, Eduard

Insulin induces a progressive increase in the resistance of subcutaneous tissue to fluid flow: Implications for insulin pump therapy

胰岛素可逐渐增加皮下组织对液体流动的阻力:对胰岛素泵治疗的启示

Regittnig, Werner; Tschaikner, Mathias; Tuca, Alexandru-Cristian; Simic, Amra; Feiel, Jürgen; Schaller-Ammann, Roland; Licht, Alexander H; Jungklaus, Miró; Pieber, Thomas R

Hedgehog and Gpr161: Regulating cAMP Signaling in the Primary Cilium

Hedgehog 和 Gpr161:调节初级纤毛中的 cAMP 信号传导

Tschaikner, Philipp; Enzler, Florian; Torres-Quesada, Omar; Aanstad, Pia; Stefan, Eduard

KinCon: Cell-based recording of full-length kinase conformations

KinCon:基于细胞的全长激酶构象记录

Enzler, Florian; Tschaikner, Philipp; Schneider, Rainer; Stefan, Eduard

Mutation-oriented profiling of autoinhibitory kinase conformations predicts RAF inhibitor efficacies

自抑制激酶构象突变导向分析可预测 RAF 抑制剂疗效

Johanna E Mayrhofer, Florian Enzler, Andreas Feichtner, Ruth Röck, Jakob Fleischmann, Andrea Raffeiner, Philipp Tschaikner, Egon Ogris, Roland G Huber, Markus Hartl, Rainer Schneider, Jakob Troppmair, Omar Torres-Quesada, Eduard Stefan

LAMTOR/Ragulator is a negative regulator of Arl8b- and BORC-dependent late endosomal positioning

LAMTOR/Ragulator 是 Arl8b 和 BORC 依赖性晚期内体定位的负调控因子。

Przemyslaw A Filipek ,Mariana E G de Araujo ,Georg F Vogel ,Cedric H De Smet ,Daniela Eberharter ,Manuele Rebsamen ,Elena L Rudashevskaya ,Leopold Kremser ,Teodor Yordanov ,Philipp Tschaikner ,Barbara G Fürnrohr ,Stefan Lechner ,Theresia Dunzendorfer-Matt ,Klaus Scheffzek ,Keiryn L Bennett ,Giulio Superti-Furga ,Herbert H Lindner ,Taras Stasyk ,Lukas A Huber

Gpr161 anchoring of PKA consolidates GPCR and cAMP signaling

Gpr161 锚定 PKA 巩固 GPCR 和 cAMP 信号传导

Verena A Bachmann, Johanna E Mayrhofer, Ronit Ilouz, Philipp Tschaikner, Philipp Raffeiner, Ruth Röck, Mathieu Courcelles, Federico Apelt, Tsan-Wen Lu, George S Baillie, Pierre Thibault, Pia Aanstad, Ulrich Stelzl, Susan S Taylor, Eduard Stefan1

In-vivo detection of binary PKA network interactions upon activation of endogenous GPCRs

体内检测内源性GPCR激活后二元PKA网络相互作用

Röck, Ruth; Bachmann, Verena; Bhang, Hyo-Eun C; Malleshaiah, Mohan; Raffeiner, Philipp; Mayrhofer, Johanna E; Tschaikner, Philipp M; Bister, Klaus; Aanstad, Pia; Pomper, Martin G; Michnick, Stephen W; Stefan, Eduard