日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

One-Pot Gateway to Quinazoline-Thiohydantoin Fused Scaffolds and Discovery of Their Antileukemic Activity

一锅法合成喹唑啉-硫代乙内酰脲稠合骨架及其抗白血病活性

Kersting, Lena; Zippel, Christoph; Herrmann, Lars; Elbadawi, Mohamed; Seo, Ean-Jeong; Heckmann, Felix; Saeed, Mohamed E M; Gaube, Angelika; Tailor, Dhanir; Dheeraj, Arpit; Malhotra, Sanjay V; Muehlich, Susanne; Efferth, Thomas; Tsogoeva, Svetlana B

Catalyzed Enantioselective Organic Synthesis

催化对映选择性有机合成

Schanze, Kirk S; Tsogoeva, Svetlana B

Organic Synthesis and Catalysis Enable Facile Access to Bioactive Compounds and Drugs

有机合成和催化技术为获取生物活性化合物和药物提供了便利

Tsogoeva, Svetlana B; Schanze, Kirk S

Development and mechanistic studies of calcium-BINOL phosphate-catalyzed hydrocyanation of hydrazones

钙-BINOL磷酸盐催化腙氢氰化反应的研制及机理研究

Tortora, Carola; Fischer, Christian Andreas; Kohlbauer, Sascha; Zamfir, Alexandru; Ballmann, Gerd M; Pahl, Jürgen; Harder, Sjoerd; Tsogoeva, Svetlana B

Access to Artemisinin-Triazole Antimalarials via Organo-Click Reaction: High In Vitro/In Vivo Activity against Multi-Drug-Resistant Malaria Parasites

通过有机点击反应合成青蒿素-三唑类抗疟药:对多重耐药疟原虫具有很高的体外/体内活性

Herrmann, Lars; Leidenberger, Maria; Quadros, Helenita C; Grau, Benedikt W; Hampel, Frank; Friedrich, Oliver; Moreira, Diogo R M; Kappes, Barbara; Tsogoeva, Svetlana B

Characterization of antimalarial activity of artemisinin-based hybrid drugs

青蒿素类杂合药物抗疟活性的表征

Quadros, Helenita Costa; Herrmann, Lars; Manaranche, Jeanne; Paloque, Lucie; Borges-Silva, Mariana C; Dziwornu, Godwin Akpeko; D'Alessandro, Sarah; Chibale, Kelly; Basilico, Nicoletta; Benoit-Vical, Françoise; Tsogoeva, Svetlana B; Moreira, Diogo Rodrigo M

Catalytic multi-step domino and one-pot reactions

催化多步多米诺反应和一锅反应

Tsogoeva, Svetlana B

Autofluorescent antimalarials by hybridization of artemisinin and coumarin: in vitro/in vivo studies and live-cell imaging

青蒿素与香豆素杂交产生的自发荧光抗疟药:体外/体内研究和活细胞成像

Herrmann, Lars; Leidenberger, Maria; Sacramento de Morais, Adrielle; Mai, Christina; Çapci, Aysun; da Cruz Borges Silva, Mariana; Plass, Fabian; Kahnt, Axel; Moreira, Diogo R M; Kappes, Barbara; Tsogoeva, Svetlana B

Front Cover: Anti‐SARS‐CoV‐2 Inhibitory Profile of New Quinoline Compounds in Cell Culture‐Based Infection Models (Chem. Eur. J. 4/2022)

封面:新型喹啉化合物在基于细胞培养的感染模型中的抗SARS-CoV-2抑制特性(Chem. Eur. J. 4/2022)

Pan, Sudip; Frenking, Gernot; Herrmann, Lars; Hahn, Friedrich; Wangen, Christina; Marschall, Manfred; Tsogoeva, Svetlana B

The Trimeric Artesunate Analog TF27, a Broadly Acting Anti-Infective Model Drug, Exerts Pronounced Anti-SARS-CoV-2 Activity Spanning Variants and Host Cell Types

三聚体青蒿琥酯类似物TF27是一种广谱抗感染模型药物,对多种SARS-CoV-2变异株和宿主细胞类型均表现出显著的抗病毒活性。

Hahn, Friedrich; Wangen, Christina; Häge, Sigrun; Herrmann, Lars; Herrmann, Alexandra; Tsogoeva, Svetlana B; Marschall, Manfred