日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Hybridization Approach Applied to Umbelliferon and Vanilloids toward New Inhibitors of Carbonic Anhydrases IX and XII with In Vitro Antiproliferative and Anti-inflammatory Activities

利用杂交方法筛选伞形酮和香草醛类化合物,以期获得具有体外抗增殖和抗炎活性的碳酸酐酶IX和XII新型抑制剂。

Melfi, Francesco; Mencarelli, Noemi; Carradori, Simone; Gallorini, Marialucia; Angeli, Andrea; Poli, Giulio; Cataldi, Amelia; D'Agostino, Ilaria; Di Credico, Andrea; Di Baldassarre, Angela; Tuccinardi, Tiziano; Supuran, Claudiu T

Novel Insights on Benzo[b]thiophene Analogues for MAO-B Inhibition and Neuroprotection: Design, Synthesis, Molecular Modelling Studies and Biological Activity

苯并[b]噻吩类似物在MAO-B抑制和神经保护方面的新见解:设计、合成、分子建模研究和生物活性

Arrighi, Francesca; Berrino, Emanuela; Guglielmi, Paolo; Carradori, Simone; Marconi, Guya Diletta; Pizzicannella, Jacopo; Guarnieri, Simone; Tuccinardi, Tiziano; Poli, Giulio; Pepi, Federico; Troiani, Anna; Salvitti, Chiara; Di Noi, Alessia; Coluccia, Michele; Buttitta, Giorgio; Pontecorvi, Virginia; Granese, Arianna; Chimenti, Paola; Secci, Daniela; Petzer, Anel; Petzer, Jacobus Petrus; Diomede, Francesca

The Burden of Obesity and Type 1 Diabetes: Distinct and Synergistic Effects to Worsen Perceived Health and Psychosocial Distress

肥胖和1型糖尿病的负担:二者对感知健康和心理社会困扰的独特和协同影响

Risi, Renata; Pauletto, Domiziana; Zanghi Buffi, Valeria; Berna, Valentina; Carafa, Andrea; Barbaro, Federica; De Vita, Francesco; D'Onofrio, Luca; Amendolara, Rocco; Lauria Pantano, Angelo; Di Flaviani, Alessandra; Zampetti, Simona; Tuccinardi, Dario; Buzzetti, Raffaella; Maddaloni, Ernesto

Development of Glycoconjugated MAGL Inhibitors with Glucose-Dependent Antiproliferative Activity

开发具有葡萄糖依赖性抗增殖活性的糖缀合MAGL抑制剂

Bononi, Giulia; Bertini, Federica; Masoni, Samuele; Stefano, Miriana Di; Mosca, Rossella; Felice, Francesca; Signore, Giovanni; Minutolo, Filippo; Granchi, Carlotta; Tuccinardi, Tiziano; Di Bussolo, Valeria

Evolving kidney disease phenotypes in type 2 diabetes: declining albuminuria and increasing isolated low eGFR

2型糖尿病肾脏疾病表型演变:白蛋白尿减少和孤立性低eGFR增加

De Cosmo, Salvatore A; Russo, Giuseppina; Nicolucci, Antonio; Rossi, Chiara; Graziano, Giusi; Fioretto, Paola; Tuccinardi, Dario; Viazzi, Francesca; Sartore, Giovanni; Muscarà, Andrea; Cuttone, Alessandro; Piscitelli, Pamela; Candido, Riccardo; Di Cianni, Graziano; Pontremoli, Roberto

Italian clinical practice GRADE-based guidelines on the diagnosis and treatment of overweight and obesity, endorsed by the Italian National Institute of Health

意大利国家卫生研究院认可的基于GRADE标准的意大利临床实践指南,用于诊断和治疗超重和肥胖。

Barazzoni, Rocco; Buscemi, Silvio; Busetto, Luca; Sbraccia, Paolo; Bo, Simona; Cereda, Emanuele; Chianelli, Marco; Chiappetta, Sonja; Dalle Grave, Riccardo; de Caro, Walter; Docimo, Giovanni; Galloro, Giuseppe; Iannone, Primiano; Leonetti, Frida; Lisso, Fabrizia; Manca, Maria Caterina; Medea, Gerardo; Merli, Manuela; Moretti, Anna Maria; Navarra, Giuseppe; Pagotto, Uberto; Paolini, Barbara; Papa, Giovanni; Perrotta, Nicola; Pession, Andrea; Pilone, Vincenzo; Provenzano, Vincenzo; Rizzo, Cecilia Ricciardi; Santomauro, Maurizio; Segura Garcia, Cristina; Spandonaro, Federico; Sukkar, Samir; Todisco, Patrizia; Tuccinardi, Dario; Vania, Andrea; Vanzi, Valentina; Williams, Riccardo; Zani, Iris; Ragghianti, Benedetta; Silverii, Giovanni Antonio; Belluzzi, Amanda; Masulli, Maria; Redini, Maddalena; Monami, Matteo

Convergent Total Synthesis of Aleutianamine

阿留申胺的汇聚合成全合成

Tuccinardi, Joseph P; Wood, John L

Convergent Total Synthesis of Erchinines A and B and Their C20 Epimers

Erchinine A 和 B 及其 C20 差向异构体的汇聚合成

Sun Cho, Yong; Tuccinardi, Joseph P; Wood, John L

Development of the First Small-Molecule Inhibitor Targeting Oncostatin M for Treatment of Breast Cancer

首个靶向抑癌素M的小分子抑制剂的研发及其在乳腺癌治疗中的应用

Cody L Wolf ,Andrea Feci ,Joseph P Tuccinardi ,Grace H Coughlin ,Kelsey A Holdaway ,Thaaer Muhammed ,Clyde Pruett ,Darren Lighter ,Cooper McGrath ,Terrell Engmann ,Maria Pou-Torres ,Brittany Rushing ,Luke Woodbury ,Sierra E Haile ,Hannah Scott ,Ken Tawara ,Simion Dinca ,Dong Xu ,Matthew D King ,Lisa Rose Warner ,Cheryl L Jorcyk ,Don L Warner

GLP-1 and GIP Beyond Glycaemia: Evolutionary Roles in Energy Optimisation and Organ Protection

GLP-1 和 GIP 超越血糖:在能量优化和器官保护中的进化作用

Tuccinardi, Dario; Watanabe, Mikiko; Masi, Davide; Gianfrilli, Daniele; Manfrini, Silvia; le Roux, Carel W