日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tonsillar Microbiome-Derived Lantibiotics Induce Structural Changes of IL-6 and IL-21 Receptors and Modulate Host Immunity

扁桃体微生物组衍生的羊毛硫抗生素诱导 IL-6 和 IL-21 受体的结构变化并调节宿主免疫

Jing Li, Jiayang Jin, Shenghui Li, Yan Zhong, Yuebo Jin, Xuan Zhang, Binbin Xia, Yinhua Zhu, Ruochun Guo, Xiaolin Sun, Jianping Guo, Fanlei Hu, Wenjing Xiao, Fei Huang, Hua Ye, Ru Li, Yunshan Zhou, Xiaohong Xiang, Haihong Yao, Qiulong Yan, Li Su, Lijun Wu, Tuoping Luo, Yudong Liu, Xiaohuan Guo, Junj

Elimination of senescent cells by β-galactosidase-targeted prodrug attenuates inflammation and restores physical function in aged mice

β-半乳糖苷酶靶向前药消除衰老细胞可减轻老年小鼠的炎症并恢复身体机能

Yusheng Cai #, Huanhuan Zhou #, Yinhua Zhu #, Qi Sun, Yin Ji, Anqi Xue, Yuting Wang, Wenhan Chen, Xiaojie Yu, Longteng Wang, Han Chen, Cheng Li, Tuoping Luo, Hongkui Deng

Structural insights into the inhibition mechanism of human sterol O-acyltransferase 1 by a competitive inhibitor

竞争性抑制剂对人类固醇 O-酰基转移酶 1 抑制机制的结构洞察

Chengcheng Guan, Yange Niu, Si-Cong Chen, Yunlu Kang, Jing-Xiang Wu, Koji Nishi, Catherine C Y Chang, Ta-Yuan Chang, Tuoping Luo, Lei Chen

A modular PROTAC design for target destruction using a degradation signal based on a single amino acid

一种使用基于单个氨基酸的降解信号进行靶标破坏的模块化 PROTAC 设计

Karthigayan Shanmugasundaram, Peng Shao, Han Chen, Bismarck Campos, Stanton F McHardy, Tuoping Luo, Hai Rao

STK33 kinase inhibitor BRD-8899 has no effect on KRAS-dependent cancer cell viability

STK33 激酶抑制剂 BRD-8899 对 KRAS 依赖性癌细胞活力无影响

Tuoping Luo, Kristina Masson, Jacob D Jaffe, Whitney Silkworth, Nathan T Ross, Christina A Scherer, Claudia Scholl, Stefan Fröhling, Steven A Carr, Andrew M Stern, Stuart L Schreiber, Todd R Golub