日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A brain-penetrant P2X7R antagonist mitigates Alzheimer's disease pathology

一种能穿透血脑屏障的P2X7R拮抗剂可减轻阿尔茨海默病病理。

Turcu, Andreea L; Oken, Adam C; Griñán-Ferré, Christian; Durner, Anna; Sierra-Marquez, Juan; Hinz-Kowalik, Sonja; Nagel, Jessica; Lee, So-Deok; Tzortzini, Efpraxia; Georgiou, Kyriakos; Bhol, Mamina; Baz, Zuriñe; Llop, Jordi; Schneider, Marion; Barbaraci, Carla; Kim, Ga-Ram; Barniol-Xicota, Marta; Val, Cristina; Brea, José; Loza, M Isabel; Pérez, Belén; Naesens, Lieve; Kolocouris, Antonios; Kim, Yong-Chul; Müller, Christa E; Nicke, Annette; Pallàs, Mercè; Mansoor, Steven E; Vázquez, Santiago

A polycyclic scaffold identified by structure-based drug design effectively inhibits the human P2X7 receptor

基于结构的药物设计鉴定出的一种多环骨架能有效抑制人P2X7受体。

Oken, Adam C; Turcu, Andreea L; Tzortzini, Eva; Georgiou, Kyriakos; Nagel, Jessica; Westermann, Franka G; Barniol-Xicota, Marta; Seidler, Jonas; Kim, Ga-Ram; Lee, So-Deok; Nicke, Annette; Kim, Yong-Chul; Müller, Christa E; Kolocouris, Antonios; Vázquez, Santiago; Mansoor, Steven E

Memantine inhibits calcium-permeable AMPA receptors.

美金刚抑制钙离子通透性AMPA受体

Carrillo Elisa, Montaño Romero Alejandra, Gonzalez Cuauhtemoc U, Turcu Andreea L, Vázquez Santiago, Twomey Edward C, Jayaraman Vasanthi

Dimethoxybenzohomoadamantane-based soluble epoxide hydrolase inhibitors: in vivo efficacy in a murine model of chemotherapy-induced neuropathic pain

基于二甲氧基苯并高金刚烷的可溶性环氧化物水解酶抑制剂:在化疗诱导神经性疼痛小鼠模型中的体内疗效

Codony, Sandra; Jora, Beatrice; Santos-Caballero, Miriam; Qiu, Qiongju; Calvó-Tusell, Carla; Escriche, Celia; Turcu, Andreea L; Prischi, Filippo; Bartra, Clara; Val, Cristina; Morisseau, Christophe; Pérez, Belén; Bertran-Mostazo, Andrea; Osuna, Sílvia; Corpas, Rubén; Griñán-Ferré, Christian; Galdeano, Carles; Loza, M Isabel; Pallàs, Mercè; Sanfeliu, Coral; Hammock, Bruce D; Brea, José; Feixas, Ferran; Conte, Maria R; Cobos, Enrique J; Vázquez, Santiago

The Tuberculosis Drug Candidate SQ109 and Its Analogs Have Multistage Activity against Plasmodium falciparum

结核病候选药物SQ109及其类似物对恶性疟原虫具有多阶段活性

Watson, Savannah J; van der Watt, Mariëtte E; Theron, Anjo; Reader, Janette; Tshabalala, Sizwe; Erlank, Erica; Koekemoer, Lizette L; Naude, Mariska; Stampolaki, Marianna; Adewole, Feyisola; Sadowska, Katie; Pérez-Lozano, Pilar; Turcu, Andreea L; Vázquez, Santiago; Ko, Jihee; Mazurek, Ben; Singh, Davinder; Malwal, Satish R; Njoroge, Mathew; Chibale, Kelly; Onajole, Oluseye K; Kolocouris, Antonios; Oldfield, Eric; Birkholtz, Lyn-Marié

Inhibition of NMDA receptors through a membrane-to-channel path

通过膜到通道途径抑制NMDA受体

Wilcox, Madeleine R; Nigam, Aparna; Glasgow, Nathan G; Narangoda, Chamali; Phillips, Matthew B; Patel, Dhilon S; Mesbahi-Vasey, Samaneh; Turcu, Andreea L; Vázquez, Santiago; Kurnikova, Maria G; Johnson, Jon W

A Novel NMDA Receptor Antagonist Protects against Cognitive Decline Presented by Senescent Mice.

一种新型 NMDA 受体拮抗剂可保护衰老小鼠免受认知能力下降的影响

Companys-Alemany Júlia, Turcu Andreea L, Bellver-Sanchis Aina, Loza Maria I, Brea José M, Canudas Anna M, Leiva Rosana, Vázquez Santiago, Pallàs Mercè, Griñán-Ferré Christian

Pharmacological and Electrophysiological Characterization of Novel NMDA Receptor Antagonists

新型NMDA受体拮抗剂的药理学和电生理学表征

Leiva, Rosana; Phillips, Matthew B; Turcu, Andreea L; Gratacòs-Batlle, Esther; León-García, Lara; Sureda, Francesc X; Soto, David; Johnson, Jon W; Vázquez, Santiago