日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of a Radiolabeled Cyclin-Dependent Kinases 4 and 6 (CDK4/6) Inhibitor for Brain and Cancer PET Imaging

开发用于脑和癌症PET成像的放射性标记细胞周期蛋白依赖性激酶4和6(CDK4/6)抑制剂

Huang, Chun-Han; Khan, Palwasha; Xu, Sulan; Cohen, Jules; Georgakis, Georgios V; Turkman, Nashaat

Design and radiosynthesis of class-IIa HDAC inhibitor with high molar activity via repositioning the (18)F-radiolabel

通过重新定位 (18)F-放射性标记,设计并放射合成具有高摩尔活性的 IIa 类 HDAC 抑制剂

Xu, Sulan; Huang, Chun-Han; Eyermann, Christopher; Georgakis, Georgios V; Turkman, Nashaat

Design, synthesis, biochemical evaluation, radiolabeling and in vivo imaging with high affinity class-IIa histone deacetylase inhibitor for molecular imaging and targeted therapy

利用高亲和力IIa类组蛋白去乙酰化酶抑制剂进行分子成像和靶向治疗的设计、合成、生化评价、放射性标记和体内成像

Turkman, Nashaat; Liu, Daxing; Pirola, Isabella

PEG(2000)-DBCO surface coating increases intracellular uptake of liposomes by breast cancer xenografts

PEG(2000)-DBCO表面涂层可增加乳腺癌异种移植瘤对脂质体的细胞内摄取

Liu, Daxing; Cohen, Jules; Turkman, Nashaat

Imaging of Sleeping Beauty-Modified CD19-Specific T Cells Expressing HSV1-Thymidine Kinase by Positron Emission Tomography

利用正电子发射断层扫描技术对表达HSV1胸苷激酶的睡美人修饰的CD19特异性T细胞进行成像

Najjar, Amer M; Manuri, Pallavi R; Olivares, Simon; Flores, Leo 2nd; Mi, Tiejuan; Huls, Helen; Shpall, Elizabeth J; Champlin, Richard E; Turkman, Nashaat; Paolillo, Vincenzo; Roszik, Jason; Rabinovich, Brian; Lee, Dean A; Alauddin, Mian; Gelovani, Juri; Cooper, Laurence J N

Novel Histone Deacetylase Class IIa Selective Substrate Radiotracers for PET Imaging of Epigenetic Regulation in the Brain

用于脑表观遗传调控PET成像的新型组蛋白去乙酰化酶IIa类选择性底物放射性示踪剂

Bonomi, Robin; Mukhopadhyay, Uday; Shavrin, Aleksandr; Yeh, Hsien-Hsien; Majhi, Anjoy; Dewage, Sajeewa W; Najjar, Amer; Lu, Xin; Cisneros, G Andrés; Tong, William P; Alauddin, Mian M; Liu, Ren-Shuan; Mangner, Thomas J; Turkman, Nashaat; Gelovani, Juri G

Synthesis and preliminary evaluation of [18F]-labeled 2-oxoquinoline derivatives for PET imaging of cannabinoid CB2 receptor

合成并初步评价[18F]标记的2-氧代喹啉衍生物用于大麻素CB2受体的PET成像

Turkman, Nashaat; Shavrin, Aleksander; Paolillo, Vincenzo; Yeh, Hsin Hsien; Flores, Leo; Soghomonian, Suren; Rabinovich, Brian; Volgin, Andrei; Gelovani, Juri; Alauddin, Mian

An investigation on stereospecific fluorination at the 2'-arabino-position of a pyrimidine nucleoside: radiosynthesis of 2'-deoxy-2'-[(18)F]fluoro-5-methyl-1-β-D-arabinofuranosyluracil

对嘧啶核苷2'-阿拉伯糖位立体选择性氟化的研究:2'-脱氧-2'-[(18)F]氟-5-甲基-1-β-D-阿拉伯呋喃糖基尿嘧啶的放射合成

Turkman, Nashaat; Paolillo, Vincenzo; Gelovani, Juri G; Alauddin, Mian M

Fluorinated cannabinoid CB2 receptor ligands: synthesis and in vitro binding characteristics of 2-oxoquinoline derivatives.

氟化大麻素 CB2 受体配体:2-氧代喹啉衍生物的合成及体外结合特性

Turkman Nashaat, Shavrin Aleksander, Ivanov Roman A, Rabinovich Brian, Volgin Andrei, Gelovani Juri G, Alauddin Mian M