日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of Dual Aurora-A and Aurora-B Degrading PROTACs for MCYN-Amplified Neuroblastoma

针对MCYN扩增型神经母细胞瘤的双重Aurora-A和Aurora-B降解PROTAC的开发

Nelson, Sydney E; Tucker, James R; Prado, Madelen G; Tierney, Lillian C; Quigley, Sarah L; Lumpkin, Andrew T; Dodd, Cayden J; Hasko, Viola; Howie, Savannah L; Aastha; Ody, Britton K; Yin, Jun; Heemstra, Jennifer M; Turlington, Mark

A Biodegradable, Polymer-Supported Oxygen Atom Transfer Reagent

一种可生物降解的聚合物负载氧原子转移试剂

Ramey, Erin E; Whitman, Elizabeth L; Buller, Cole E; Tucker, James R; Jolly, Charles S; Oberle, Kjersti G; Becksvoort, Austin J; Turlington, Mark; Turlington, Christopher R

Computational Exploration of Potential CFTR Binding Sites for Type I Corrector Drugs

利用计算方法探索I型矫正药物潜在的CFTR结合位点

Lester, Anna; Sandman, Madeline; Herring, Caitlin; Girard, Christian; Dixon, Brandon; Ramsdell, Havanna; Reber, Callista; Poulos, Jack; Mitchell, Alexis; Spinney, Allison; Henager, Marissa E; Evans, Claudia N; Turlington, Mark; Johnson, Quentin R

Linkage-Specific Synthesis of Di-ubiquitin Probes Enabled by the Incorporation of Unnatural Amino Acid ThzK

引入非天然氨基酸ThzK可实现二泛素探针的连接特异性合成

Zhou, Han; Carpenter, Tomaya; Fu, Xuan; Jin, Bo; Ody, Britton; Hassan, Mohammad Sazid; Jacobs, Savannah E; Cheung, Jenny; Nicholson, Eve M; Turlington, Mark; Zhao, Bo; Lorenz, Sonja; Cropp, T Ashton; Yin, Jun

Acyl dihydropyrazolo[1,5-a]pyrimidinones as metabotropic glutamate receptor 5 positive allosteric modulators

酰基二氢吡唑并[1,5-a]嘧啶酮作为代谢型谷氨酸受体5正向变构调节剂

Malosh, Chrysa; Turlington, Mark; Bridges, Thomas M; Rook, Jerri M; Noetzel, Meredith J; Vinson, Paige N; Steckler, Thomas; Lavreysen, Hilde; Mackie, Claire; Bartolomé-Nebreda, José M; Conde-Ceide, Susana; Martínez-Viturro, Carlos M; Piedrafita, María; Sánchez-Casado, M Rosa; Macdonald, Gregor J; Daniels, J Scott; Jones, Carrie K; Niswender, Colleen M; Conn, P Jeffrey; Lindsley, Craig W; Stauffer, Shaun R

Tetrahydronaphthyridine and dihydronaphthyridinone ethers as positive allosteric modulators of the metabotropic glutamate receptor 5 (mGlu₠).

四氢萘啶和二氢萘啶酮醚作为代谢型谷氨酸受体 5 (mGluâ‚) 的正向变构调节剂

Turlington Mark, Malosh Chrysa, Jacobs Jon, Manka Jason T, Noetzel Meredith J, Vinson Paige N, Jadhav Satyawan, Herman Elizabeth J, Lavreysen Hilde, Mackie Claire, Bartolomé-Nebreda José M, Conde-Ceide Susana, Martín-Martín M Luz, Tong Han Min, López Silvia, MacDonald Gregor J, Steckler Thomas, Daniels J Scott, Weaver C David, Niswender Colleen M, Jones Carrie K, Conn P Jeffrey, Lindsley Craig W, Stauffer Shaun R

Discovery and SAR of a novel series of metabotropic glutamate receptor 5 positive allosteric modulators with high ligand efficiency

发现并研究了一系列新型代谢型谷氨酸受体5正向变构调节剂的构效关系及其配体效率

Turlington, Mark; Noetzel, Meredith J; Bridges, Thomas M; Vinson, Paige N; Steckler, Thomas; Lavreysen, Hilde; Mackie, Claire; Bartolomé-Nebreda, José M; Conde-Ceide, Susana; Tong, Han Min; Macdonald, Gregor J; Daniels, J Scott; Jones, Carrie K; Niswender, Colleen M; Conn, P Jeffrey; Lindsley, Craig W; Stauffer, Shaun R