日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of BBO-8520, a First-In-Class Direct and Covalent Dual Inhibitor of GTP-Bound (ON) and GDP-Bound (OFF) KRASG12C.

发现 BBO-8520,一种首创的直接共价双重抑制剂,可抑制 GTP 结合 (ON) 和 GDP 结合 (OFF) 的 KRASG12C

Maciag Anna E, Stice James P, Wang Bin, Sharma Alok K, Chan Albert H, Lin Ken, Singh Devansh, Dyba Marcin, Yang Yue, Setoodeh Saman, Smith Brian P, Ju Jin Hyun, Jeknic Stevan, Rabara Dana, Zhang Zuhui, Larsen Erik K, Esposito Dominic, Denson John-Paul, Ranieri Michela, Meynardie Mary, Mehdizadeh Sadaf, Alexander Patrick A, Abreu Blanco Maria, Turner David M, Xu Rui, Lightstone Felice C, Wong Kwok-Kin, Stephen Andrew G, Wang Keshi, Simanshu Dhirendra K, Sinkevicius Kerstin W, Nissley Dwight V, Wallace Eli, McCormick Frank, Beltran Pedro J

Structural insights into isoform-specific RAS-PI3Kα interactions and the role of RAS in PI3Kα activation.

从结构角度深入了解 RAS-PI3Kα 同工型特异性相互作用以及 RAS 在 PI3Kα 激活中的作用

Czyzyk Daniel, Yan Wupeng, Messing Simon, Gillette William, Tsuji Takashi, Yamaguchi Mitsuhiro, Furuzono Shinji, Turner David M, Esposito Dominic, Nissley Dwight V, McCormick Frank, Simanshu Dhirendra K

Blocking C-terminal processing of KRAS4b via a direct covalent attack on the CaaX-box cysteine.

通过对 CaaX 盒半胱氨酸进行直接共价攻击,阻断 KRAS4b 的 C 端加工

Maciag Anna E, Yang Yue, Sharma Alok K, Turner David M, DeHart Caroline J, Abdelkarim Hazem, Fan Lixin, Smith Brian P, Kumari Vandana, Dyba Marcin, Rigby Megan, Castillo Badillo Jean A, Adams Lauren, Fornelli Luca, Fox Stephen, Brafman Alla, Turbyville Thomas, Gillette William, Messing Simon, Agamasu Constance, Wolfe Andrew L, Gysin Stephan, Chan Albert H, Simanshu Dhirendra K, Esposito Dominic, Chertov Oleg, Stephen Andrew G, Arkin Michelle, Renslo Adam, Kelleher Neil L, Gaponenko Vadim, Lightstone Felice C, Nissley Dwight V, McCormick Frank

COVID-19 and algorithmic medical ethics: A Christian perspective

新冠疫情与算法医疗伦理:基督教视角

Pereira, Talmo D; Tabris, Nathaniel; Matsliah, Arie; Turner, David M; Li, Junyu; Ravindranath, Shruthi; Papadoyannis, Eleni S; Normand, Edna; Deutsch, David S; Wang, Z Yan; McKenzie-Smith, Grace C; Mitelut, Catalin C; Castro, Marielisa Diez; D'Uva, John; Kislin, Mikhail; Sanes, Dan H; Kocher, Sarah D; Wang, Samuel S-H; Falkner, Annegret L; Shaevitz, Joshua W; Murthy, Mala; Childs, Brian H

Nitinol Release of Nickel under Physiological Conditions: Effects of Surface Oxide, pH, Hydrogen Peroxide, and Sodium Hypochlorite

生理条件下镍钛合金镍的释放:表面氧化物、pH、过氧化氢和次氯酸钠的影响

Eric M Sussman, Huiyu Shi, Paul A Turner, David M Saylor, Jason D Weaver, David D Simon, Pavel Takmakov, Shiril Sivan, Hainsworth Y Shin, Matthew A Di Prima, Dianne E Godar

Rapid GMP-Compliant Expansion of SARS-CoV-2-Specific T Cells From Convalescent Donors for Use as an Allogeneic Cell Therapy for COVID-19

快速扩增符合GMP规范的SARS-CoV-2特异性T细胞(来自康复者供体),用于COVID-19的同种异体细胞疗法

Cooper, Rachel S; Fraser, Alasdair R; Smith, Linda; Burgoyne, Paul; Imlach, Stuart N; Jarvis, Lisa M; Turner, David M; Zahra, Sharon; Turner, Marc L; Campbell, John D M

The Impact of Withdrawal of Maintenance Immunosuppression and Graft Nephrectomy on HLA Sensitization and Calculated Chance of Future Transplant

停用维持性免疫抑制剂和移植肾切除术对HLA致敏及未来移植几率的影响

Nimmo, Ailish M S A; McIntyre, Sophie; Turner, David M; Henderson, Lorna K; Battle, Richard K

Targeting Non-Catalytic Cysteine Residues Through Structure-Guided Drug Discovery

通过结构导向的药物发现靶向非催化半胱氨酸残基

Hallenbeck, Kenneth K; Turner, David M; Renslo, Adam R; Arkin, Michelle R

Establishment and operation of a Good Manufacturing Practice-compliant allogeneic Epstein-Barr virus (EBV)-specific cytotoxic cell bank for the treatment of EBV-associated lymphoproliferative disease

建立并运营符合良好生产规范的同种异体EB病毒(EBV)特异性细胞毒性细胞库,用于治疗EBV相关淋巴增生性疾病

Vickers, Mark A; Wilkie, Gwen M; Robinson, Nicolas; Rivera, Nadja; Haque, Tanzina; Crawford, Dorothy H; Barry, Jacqueline; Fraser, Neil; Turner, David M; Robertson, Victoria; Dyer, Phil; Flanagan, Peter; Newlands, Helen R; Campbell, John; Turner, Marc L