A 3-(4-nitronaphthen-1-yl) amino-benzoate analog as a bifunctional AKR1C3 inhibitor and AR antagonist: Head to head comparison with other advanced AKR1C3 targeted therapeutics
3-(4-硝基萘-1-基)氨基苯甲酸酯类似物作为双功能 AKR1C3 抑制剂和 AR 拮抗剂:与其他先进的 AKR1C3 靶向疗法进行正面比较
期刊:Journal of Steroid Biochemistry and Molecular Biology
影响因子:2.7
doi:10.1016/j.jsbmb.2019.01.001
Phumvadee Wangtrakuldee, Adegoke O Adeniji, Tianzhu Zang, Ling Duan, Buddha Khatri, Barry M Twenter, Michelle A Estrada, Tyler F Higgins, Jeffrey D Winkler, Trevor M Penning