WRN structural flexibility showcased through fragment-based lead discovery of inhibitors
通过基于片段的抑制剂先导化合物发现,展现了WRN结构的灵活性
期刊:Nature Communications
影响因子:15.7
doi:10.1038/s41467-025-66768-8
Palte, Rachel L; Mandal, Mihir; Sikorska, Justyna; Villafania, Artjohn B; Rickard, Meredith M; Bauer, Robert J; Buevich, Alexei V; Chai, Xiaomei; He, Jiafang; Hussain, Zahid; Koglin, Markus; MacDonald, Hannah B; Mansueto, My S; Maskos, Klaus; Methot, Joey L; Robustelli, Jaclyn; Soriano, Aileen; Tauchert, Marcel J; Tyagarajan, Sriram; Zhang, Minjia; Klein, Daniel J; Hicks, Jacqueline D; McLaren, David G; Gabelli, Sandra B; Wyss, Daniel F