日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus MPro inhibitors with potent in vivo efficacy

基于结构的、具有高效体内疗效的高生物利用度、共价、广谱冠状病毒MPro抑制剂的发现

Tyler C Detomasi ,Gilles Degotte ,Sijie Huang ,Rahul K Suryawanshi ,Amy Diallo ,Luca Lizzadro ,Francisco J Zapatero-Belinchón ,Taha Y Taha ,Jiapeng Li ,Alicia L Richards ,Eric R Hantz ,Zain Alam ,Mauricio Montano ,Maria McCavitt-Malvido ,Rajesh Gumpena ,James R Partridge ,Galen J Correy ,Yusuke Matsui ,Annemarie F Charvat ,Isabella S Glenn ,Julia Rosecrans ,Jezrael L Revalde ,Dashiell Anderson ,Judd F Hultquist ,Michelle R Arkin ,R Jeffrey Neitz ,Danielle L Swaney ,Nevan J Krogan ,Brian K Shoichet ,Kliment A Verba ,Melanie Ott ,Adam R Renslo ,Charles S Craik

Large library docking for novel SARS-CoV-2 main protease non-covalent and covalent inhibitors

新型 SARS-CoV-2 主蛋白酶非共价和共价抑制剂的大型文库对接

Elissa A Fink, Conner Bardine, Stefan Gahbauer, Isha Singh, Tyler C Detomasi, Kris White, Shuo Gu, Xiaobo Wan, Jun Chen, Beatrice Ary, Isabella Glenn, Joseph O'Connell, Henry O'Donnell, Pavla Fajtová, Jiankun Lyu, Seth Vigneron, Nicholas J Young, Ivan S Kondratov, Arghavan Alisoltani, Lacy M Simons,

Proteases influence colony aggregation behavior in Vibrio cholerae

蛋白酶影响霍乱弧菌的菌落聚集行为

Tyler C Detomasi, Allison E Batka, Julie S Valastyan, Molly A Hydorn, Charles S Craik, Bonnie L Bassler, Michael A Marletta

Characterization of a unique polysaccharide monooxygenase from the plant pathogen Magnaporthe oryzae

植物病原菌稻瘟病菌中一种独特的多糖单加氧酶的表征

Alejandra Martinez-D'Alto, Xia Yan, Tyler C Detomasi, Richard I Sayler, William C Thomas, Nicholas J Talbot, Michael A Marletta

A Prototype Assay Multiplexing SARS-CoV-2 3CL-Protease and Angiotensin-Converting Enzyme 2 for Saliva-Based Diagnostics in COVID-19

一种多路复用 SARS-CoV-2 3CL-蛋白酶和血管紧张素转换酶 2 的原型检测方法,用于基于唾液的 COVID-19 诊断

Vallabh Suresh, Daniel A Sheik, Tyler C Detomasi, Tianqi Zhao, Theresa Zepeda, Shyam Saladi, Ummadisetti Chinna Rajesh, Kaleb Byers, Charles S Craik, Vincent Jo Davisson

A moonlighting function of a chitin polysaccharide monooxygenase, CWR-1, in Neurospora crassa allorecognition

几丁质多糖单加氧酶 CWR-1 在粗糙脉孢菌同种识别中的兼职功能

Tyler C Detomasi #, Adriana M Rico-Ramírez #, Richard I Sayler, A Pedro Gonçalves, Michael A Marletta, N Louise Glass

Substrate selectivity in starch polysaccharide monooxygenases

淀粉多糖单加氧酶的底物选择性

Van V Vu, John A Hangasky, Tyler C Detomasi, Skylar J W Henry, Son Tung Ngo, Elise A Span, Michael A Marletta

A Modular Ionophore Platform for Liver-Directed Copper Supplementation in Cells and Animals

用于细胞和动物肝脏铜补充的模块化离子载体平台

Timothy A Su, Diyala S Shihadih, Wendy Cao, Tyler C Detomasi, Marie C Heffern, Shang Jia, Andreas Stahl, Christopher J Chang