日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, synthesis, and anticancer activity of novel isocryptolepine 'aza' type acyl thiourea derivatives via combined experimental and computational approach

通过实验和计算相结合的方法设计、合成新型异隐花碱“氮杂”型酰基硫脲衍生物及其抗癌活性

Fayyaz, Ammara; Ejaz, Syeda Abida; Ahmed, Atteeque; Channar, Pervaiz Ali; Afzal, Saira; Ujan, Rabail; Saeed, Aamer; Bibi, Rifhat; Alsfouk, Bshra A; Abbas, Qamar; Sahito, Reshma; Bolte, Michael; Hökelek, Tuncer

Exploration of newly synthesized azo-thiohydantoins as the potential alkaline phosphatase inhibitors via advanced biochemical characterization and molecular modeling approaches

通过先进的生化表征和分子建模方法探索新合成的偶氮硫代乙内酰脲作为潜在的碱性磷酸酶抑制剂

Hafiz Muhammad Attaullah, Syeda Abida Ejaz, Pervaiz Ali Channar, Aamer Saeed, Rabail Ujan, Seema Zargar, Sajid Ali Channar, Reshma Sahito, Tanveer A Wani, Qamar Abbas

Dietary Effect of Withania somnifera Root Powder on Growth, Hematobiochemical Parameters, Immunity, and Disease Resistance to Aeromonas hydrophila in Cyprinus carpio

南非醉茄根粉对鲤鱼生长、血液生化指标、免疫力和对嗜水气单胞菌的抗病性的影响

Habib, Syed Sikandar; Saeed, Muhammad Qamar; Masud, Samrah; Kesbiç, Osman Sabri; Ujan, Javed Ahmed; Cravana, Cristina; Al-Rejaie, Salim S; Mohany, Mohamed; Fazio, Francesco

Identification of dimethyl 2,2'-((methylenebis(2-(2H-benzo[d][1,2,3]triazol-2-yl)-4-(2,4,4-trimethylpentan-2-yl)-6,1phenylene))bis(oxy))diacetate (TAJ4) as antagonist of NEK-Family: a future for potential drug discovery

二甲基 2,2'-((亚甲基双(2-(2H-苯并[d][1,2,3]三唑-2-基)-4-(2,4,4-三甲基戊-2-基)-6,1-亚苯基))双(氧))二乙酸酯 (TAJ4) 被鉴定为 NEK 家族拮抗剂:潜在药物发现的未来

Aziz, Mubashir; Ejaz, Syeda Abida; Channar, Pervaiz Ali; Alkhathami, Ali G; Qadri, Tahir; Hussain, Zahid; Hussaain, Mumtaz; Ujan, Rabail

Synthesis, DFT and molecular docking of novel (Z)-4-bromo-N-(4-butyl-3 (quinolin-3-yl)thiazol-2(3H)-ylidene)benzamide as elastase inhibitor

新型(Z)-4-溴-N-(4-丁基-3-(喹啉-3-基)噻唑-2(3H)-亚基)苯甲酰胺作为弹性蛋白酶抑制剂的合成、DFT计算和分子对接

Mustafa, Muhammad Naeem; Channar, Pervaiz Ali; Ejaz, Syeda Abida; Afzal, Saira; Aziz, Mubashir; Shamim, Tahira; Saeed, Aamer; Alsfouk, Aisha A; Ujan, Rabail; Abbas, Qamar; Hökelek, Tuncer

Synthesis, biological evaluation and in silico investigations of benzotriazole derivatives as potential inhibitors of NIMA related kinase

苯并三唑衍生物作为NIMA相关激酶潜在抑制剂的合成、生物学评价和计算机模拟研究

Qadri, Tahir; Aziz, Mubashir; Channar, Pervaiz Ali; Ejaz, Syeda Abida; Hussain, Mumtaz; Attaullah, Hafiz Muhammad; Ujan, Rabail; Hussain, Zahid; Zehra, Tasneem; Saeed, Aamer; Shah, M R; Ogaly, Hanan A; Al-Zahrani, Fatimah A M

Deciphering key genes involved in cisplatin resistance in kidney renal clear cell carcinoma through a combined in silico and in vitro approach

通过计算机和体外相结合的方法揭示肾透明细胞癌顺铂耐药性的关键基因

Muneeba Malik, Mamoona Maqbool, Tooba Nisar, Tazeem Akhter, Javed Ahmed Ujan, Alanood S Algarni, Fakhria A Al Joufi, Sultan Shafi K Alanazi, Mohammad Hadi Almotared, Mounir M Salem Bekhit, Muhammad Jamil

Exploring 2-Tetradecanoylimino-3-aryl-4-methyl-1,3-thiazolines Derivatives as Alkaline Phosphatase Inhibitors: Biochemical Evaluation and Computational Analysis

探索2-十四烷酰亚氨基-3-芳基-4-甲基-1,3-噻唑啉衍生物作为碱性磷酸酶抑制剂:生化评价和计算分析

Ahmed, Aftab; Rehman, Sajid-Ur; Ejaz, Syeda Abida; Saeed, Aamer; Ujan, Rabail; Channar, Pervaiz Ali; Mahar, Khalida; Sahito, Reshma; Albogami, Sarah M; Abbas, Qamar; Alorabi, Mohammed; Waard, Michel De; Batiha, Gaber El-Saber

In-silico Investigations of quinine and quinidine as potential Inhibitors of AKR1B1 and AKR1B10: Functional and structural characterization

利用计算机模拟研究奎宁和奎尼丁作为AKR1B1和AKR1B10潜在抑制剂的功能和结构表征

Ejaz, Syeda Abida; Saeed, Amna; Birmani, Pervez Rashid; Katubi, Khadijah Mohammedsalaeh; Elqahtani, Zainab Mufarreh; Al-Buriahi, M S; Ujan, Rabail; Siddique, Farhan; Ahmed, Samia Ben; Alrowaili, Z A

Synthesis, X-ray crystal structure elucidation and Hirshfeld surface analysis of N-((4-(1 H-benzo[ d]imidazole-2-yl)phenyl)carbamothioyl)benzamide: investigations for elastase inhibition, antioxidant and DNA binding potentials for biological applications

N-((4-(1 H-苯并[ d]咪唑-2-基)苯基)氨基硫酰基)苯甲酰胺的合成、X 射线晶体结构解析和 Hirshfeld 表面分析:研究其对弹性蛋白酶的抑制作用、抗氧化作用和 DNA 结合潜力,用于生物应用

Nasima Arshad, Mamoona Rafiq, Rabail Ujan, Aamer Saeed, Shahid I Farooqi, Fouzia Perveen, Pervaiz Ali Channar, Saba Ashraf, Qamar Abbas, Ashfaq Ahmed, Tuncer Hokelek, Manpreet Kaur, Jerry P Jasinski