日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Combining BET inhibition with SMAC mimetics restricts tumor growth and triggers immune surveillance in preclinical cancer models

在临床前癌症模型中,BET抑制剂与SMAC模拟物联合使用可抑制肿瘤生长并触发免疫监视。

Ksenija Slavic Obradovic ,Florian Ebner ,Artem V Artemov ,Martina Miotto ,Paula-Elena Traexler ,Robin Jacob ,Ha Pham Thi Thanh ,Regina Ruzicka ,Andreas Wernitznig ,Ines Baumann ,Daniel Gerlach ,Maria-Antonietta Impagnatiello ,Salvatore Siena ,Mary Murphy ,Reniqua House ,Ulrich Reiser ,Valeria Santoro ,Johannes Popow ,Sebastian Carotta ,Anke Baum ,Jesse Lipp ,Alberto Bardelli ,Ulrike Tontsch-Grunt ,Mariangela Russo ,Martin Aichinger

Tumor microenvironment mimicking 3D models unveil the multifaceted effects of SMAC mimetics

模拟肿瘤微环境的3D模型揭示了SMAC模拟物的多方面作用

Catarina Pinto,Ksenija Slavic-Obradovic,Daniela Fürweger,Barbara Thaler,Abdallah Souabni,Sebastian Carotta,Martin Aichinger,Ulrich Reiser,Maria Antonietta Impagnatiello,Iñigo Tirapu

Fragment-based discovery of a chemical probe for the PWWP1 domain of NSD3

基于片段的 NSD3 PWWP1 结构域化学探针的发现

Jark Böttcher, David Dilworth, Ulrich Reiser, Ralph A Neumüller, Michael Schleicher, Mark Petronczki, Markus Zeeb, Nikolai Mischerikow, Abdellah Allali-Hassani, Magdalena M Szewczyk, Fengling Li, Steven Kennedy, Masoud Vedadi, Dalia Barsyte-Lovejoy, Peter J Brown, Kilian V M Huber, Catherine M Roger