日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

NRX-0492 degrades wild-type and C481 mutant BTK and demonstrates in vivo activity in CLL patient-derived xenografts

NRX-0492 可降解野生型和 C481 突变型 BTK,并在 CLL 患者来源的异种移植模型中显示出体内活性。

Deyi Zhang ,Hailey M Harris ,Jonathan Chen ,Jen Judy ,Gabriella James ,Aileen Kelly ,Joel McIntosh ,Austin Tenn-McClellan ,Eileen Ambing ,Ying Siow Tan ,Hao Lu ,Stefan Gajewski ,Matthew C Clifton ,Stephanie Yung ,Daniel W Robbins ,Mehdi Pirooznia ,Sigrid S Skånland ,Erika Gaglione ,Maissa Mhibik ,Chingiz Underbayev ,Inhye E Ahn ,Clare Sun ,Sarah E M Herman ,Mark Noviski ,Adrian Wiestner

CD49d Expression Identifies a Biologically Distinct Subtype of Chronic Lymphocytic Leukemia with Inferior Progression-Free Survival on BTK Inhibitor Therapy

CD49d表达可识别出一种生物学上独特的慢性淋巴细胞白血病亚型,该亚型在接受BTK抑制剂治疗后无进展生存期较差。

Alsadhan, Anfal; Chen, Jonathan; Gaglione, Erika M; Underbayev, Chingiz; Tuma, Pamela L; Tian, Xin; Freeman, Lita A; Baskar, Sivasubramanian; Nierman, Pia; Soto, Susan; Itsara, Andy; Ahn, Inhye E; Sun, Clare; Bibikova, Elena; Hartmann, Tanja Nicole; Mhibik, Maissa; Wiestner, Adrian

MARCKS affects cell motility and response to BTK inhibitors in CLL

MARCKS 影响 CLL 中的细胞迁移和对 BTK 抑制剂的反应

Laura Beckmann, Valeska Berg, Clarissa Dickhut, Clare Sun, Olaf Merkel, Johannes Bloehdorn, Sandra Robrecht, Marc Seifert, Alexandra da Palma Guerreiro, Julia Claasen, Stefan Loroch, Matteo Oliverio, Chingiz Underbayev, Lauren Vaughn, Daniel Thomalla, Malte F Hülsemann, Eugen Tausch, Kirsten Fischer

IKAP-Identifying K mAjor cell Population groups in single-cell RNA-sequencing analysis

IKAP——在单细胞RNA测序分析中识别K mA主要细胞群

Chen, Yun-Ching; Suresh, Abhilash; Underbayev, Chingiz; Sun, Clare; Singh, Komudi; Seifuddin, Fayaz; Wiestner, Adrian; Pirooznia, Mehdi

A CD19/CD3 bispecific antibody for effective immunotherapy of chronic lymphocytic leukemia in the ibrutinib era

在伊布替尼时代,一种用于有效治疗慢性淋巴细胞白血病的CD19/CD3双特异性抗体

Robinson, Hannah R; Qi, Junpeng; Cook, Erika M; Nichols, Cydney; Dadashian, Eman L; Underbayev, Chingiz; Herman, Sarah E M; Saba, Nakhle S; Keyvanfar, Keyvan; Sun, Clare; Ahn, Inhye E; Baskar, Sivasubramanian; Rader, Christoph; Wiestner, Adrian

Clonal evolution leading to ibrutinib resistance in chronic lymphocytic leukemia

慢性淋巴细胞白血病中导致伊布替尼耐药性的克隆演化

Ahn, Inhye E; Underbayev, Chingiz; Albitar, Adam; Herman, Sarah E M; Tian, Xin; Maric, Irina; Arthur, Diane C; Wake, Laura; Pittaluga, Stefania; Yuan, Constance M; Stetler-Stevenson, Maryalice; Soto, Susan; Valdez, Janet; Nierman, Pia; Lotter, Jennifer; Xi, Liqiang; Raffeld, Mark; Farooqui, Mohammed; Albitar, Maher; Wiestner, Adrian

MALT1 Inhibition Is Efficacious in Both Naïve and Ibrutinib-Resistant Chronic Lymphocytic Leukemia.

MALT1抑制剂对原发性和伊布替尼耐药的慢性淋巴细胞白血病均有效

Saba Nakhle S, Wong Deanna H, Tanios Georges, Iyer Jessica R, Lobelle-Rich Patricia, Dadashian Eman L, Liu Delong, Fontan Lorena, Flemington Erik K, Nichols Cydney M, Underbayev Chingiz, Safah Hana, Melnick Ari, Wiestner Adrian, Herman Sarah E M

The evolutionary landscape of chronic lymphocytic leukemia treated with ibrutinib targeted therapy

伊布替尼靶向治疗慢性淋巴细胞白血病的演变图景

Landau, Dan A; Sun, Clare; Rosebrock, Daniel; Herman, Sarah E M; Fein, Joshua; Sivina, Mariela; Underbayev, Chingiz; Liu, Delong; Hoellenriegel, Julia; Ravichandran, Sarangan; Farooqui, Mohammed Z H; Zhang, Wandi; Cibulskis, Carrie; Zviran, Asaf; Neuberg, Donna S; Livitz, Dimitri; Bozic, Ivana; Leshchiner, Ignaty; Getz, Gad; Burger, Jan A; Wiestner, Adrian; Wu, Catherine J

Pathogenic role of B-cell receptor signaling and canonical NF-κB activation in mantle cell lymphoma.

B 细胞受体信号传导和经典 NF-κB 激活在套细胞淋巴瘤中的致病作用

Saba Nakhle S, Liu Delong, Herman Sarah E M, Underbayev Chingiz, Tian Xin, Behrend David, Weniger Marc A, Skarzynski Martin, Gyamfi Jennifer, Fontan Lorena, Melnick Ari, Grant Cliona, Roschewski Mark, Navarro Alba, Beà Sílvia, Pittaluga Stefania, Dunleavy Kieron, Wilson Wyndham H, Wiestner Adrian

Role of mir-15a/16-1 in early B cell development in a mouse model of chronic lymphocytic leukemia

mir-15a/16-1 在慢性淋巴细胞白血病小鼠模型中早期 B 细胞发育中的作用

Chingiz Underbayev, Siddha Kasar, William Ruezinsky, Heba Degheidy, Joel Solomon Schneider, Gerald Marti, Steven R Bauer, Diego Fraidenraich, Marilyn M Lightfoote, Vijay Parashar, Elizabeth Raveche, Mona Batish