日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural insights into chemoresistance mutants of BCL-2 and their targeting by stapled BAD BH3 helices.

BCL-2 化学耐药突变体的结构见解及其被 BAD BH3 螺旋钉合物靶向的作用。

DeAngelo Thomas M, Adhikary Utsarga, Korshavn Kyle J, Seo Hyuk-Soo, Brotzen-Smith Clara R, Camara Christina M, Dhe-Paganon Sirano, Bird Gregory H, Wales Thomas E, Walensky Loren D

A triple-action PROTAC for wild-type p53 cancer therapy

用于野生型p53癌症治疗的三重作用PROTAC

Bird, Gregory H; Adhikary, Utsarga; Schmidt, Michael J; Godes, Marina; Tesar, Bethany; Camara, Christina M; Paulo, Joao A; Vidlak, Julia F; DeAngelo, Thomas M; Marquez, Marilyn; Gokhale, Prafulla; Li, Ruitong; Ho Sui, Shannan J; Cameron, Michael D; Gygi, Steven P; Walensky, Loren D

Covalent inhibition of pro-apoptotic BAX.

共价抑制促凋亡蛋白BAX

McHenry Matthew W, Shi Peiwen, Camara Christina M, Cohen Daniel T, Rettenmaier T Justin, Adhikary Utsarga, Gygi Micah A, Yang Ka, Gygi Steven P, Wales Thomas E, Engen John R, Wells James A, Walensky Loren D

Targeting MCL-1 triggers DNA damage and an anti-proliferative response independent from apoptosis induction

靶向MCL-1可引发DNA损伤和抗增殖反应,且该反应独立于细胞凋亡诱导。

Utsarga Adhikary ,Joao A Paulo ,Marina Godes ,Shrabasti Roychoudhury ,Michelle S Prew ,Yael Ben-Nun ,Ellen W Yu ,Amit Budhraja ,Joseph T Opferman ,Dipanjan Chowdhury ,Steven P Gygi ,Loren D Walensky

MCL-1 is a master regulator of cancer dependency on fatty acid oxidation

MCL-1是癌症对脂肪酸氧化依赖性的关键调控因子。

Michelle S Prew ,Utsarga Adhikary ,Dong Wook Choi ,Erika P Portero ,Joao A Paulo ,Pruthvi Gowda ,Amit Budhraja ,Joseph T Opferman ,Steven P Gygi ,Nika N Danial ,Loren D Walensky

Targeting a helix-in-groove interaction between E1 and E2 blocks ubiquitin transfer

靶向 E1 和 E2 之间的螺旋槽相互作用可阻断泛素转移

Ann M Cathcart, Gregory H Bird, Thomas E Wales, Henry D Herce, Edward P Harvey, Zachary J Hauseman, Catherine E Newman, Utsarga Adhikary, Michelle S Prew, Tun Oo, Susan Lee, John R Engen, Loren D Walensky

Radiation therapy primes tumors for nanotherapeutic delivery via macrophage-mediated vascular bursts

放射疗法通过巨噬细胞介导的血管破裂,使肿瘤更容易接受纳米治疗药物的递送。

Miller, Miles A; Chandra, Ravi; Cuccarese, Michael F; Pfirschke, Christina; Engblom, Camilla; Stapleton, Shawn; Adhikary, Utsarga; Kohler, Rainer H; Mohan, James F; Pittet, Mikael J; Weissleder, Ralph

Contributions of vulnerable hydrogeomorphic habitats to endemic plant diversity on the Kas Plateau, Western Ghats

脆弱水文地貌生境对西高止山脉卡斯高原特有植物多样性的贡献

Bhattarai, Utsarga; Tetali, Pundarikakshudu; Kelso, Sylvia