日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimizing uPAR-targeting radiopeptides for improved tissue distribution: progress towards radionuclide therapy

优化靶向 uPAR 的放射性肽以改善组织分布:放射性核素治疗的进展

Vaccarin, Christian; Beyer, Darja; Schmid, Jerome V; Klein, Bastian; Jegathasan, Jathursa; Behera, Shreshtha; Deupi, Xavier; Schibli, Roger; Müller, Cristina

Development of lisinopril radioconjugates for nuclear imaging of the angiotensin converting enzyme

赖诺普利放射性偶联物在血管紧张素转换酶核成像中的应用研究

Vaccarin, Christian; Beyer, Darja; Moiseeva, Anzhelika; Favaretto, Chiara; van der Meulen, Nicholas P; Hunkeler, Benjamin D; Rupp, Niels J; Marzaro, Giovanni; Schibli, Roger; Müller, Cristina

Design and Preclinical Evaluation of Novel uPAR-Targeting Radiopeptides Modified with an Albumin-Binding Entity

利用白蛋白结合实体修饰的新型uPAR靶向放射性肽的设计和临床前评估

Beyer, Darja; Vaccarin, Christian; Schmid, Jerome V; Deberle, Luisa M; Deupi, Xavier; Schibli, Roger; Müller, Cristina

Development of radiofluorinated MLN-4760 derivatives for PET imaging of the SARS-CoV-2 entry receptor ACE2

开发用于SARS-CoV-2进入受体ACE2 PET成像的放射性氟化MLN-4760衍生物

Wang, Jinling; Beyer, Darja; Vaccarin, Christian; He, Yingfang; Tanriver, Matthias; Benoit, Roger; Deupi, Xavier; Mu, Linjing; Bode, Jeffrey W; Schibli, Roger; Müller, Cristina

Design and Preclinical Evaluation of a Novel Prostate-Specific Membrane Antigen Radioligand Modified with a Transthyretin Binder.

设计和临床前评估一种新型前列腺特异性膜抗原放射性配体,该配体经转甲状腺素结合剂修饰

Vaccarin Christian, Mapanao Ana Katrina, Deberle Luisa M, Becker Anna E, Borgna Francesca, Marzaro Giovanni, Schibli Roger, Müller Cristina

Investigations Using Albumin Binders to Modify the Tissue Distribution Profile of Radiopharmaceuticals Exemplified with Folate Radioconjugates

利用白蛋白结合剂改变放射性药物组织分布特征的研究——以叶酸放射性偶联物为例

Busslinger, Sarah D; Becker, Anna E; Vaccarin, Christian; Deberle, Luisa M; Renz, Marie-Luise; Groehn, Viola; Schibli, Roger; Müller, Cristina

A tool for nuclear imaging of the SARS-CoV-2 entry receptor: molecular model and preclinical development of ACE2-selective radiopeptides

SARS-CoV-2 进入受体的核成像工具:ACE2 选择性放射性肽的分子模型和临床前开发

Darja Beyer #, Christian Vaccarin #, Xavier Deupi, Ana Katrina Mapanao, Susan Cohrs, Fan Sozzi-Guo, Pascal V Grundler, Nicholas P van der Meulen, Jinling Wang, Matthias Tanriver, Jeffrey W Bode, Roger Schibli, Cristina Müller

Self-Emulsifying Formulations to Increase the Oral Bioavailability of 4,6,4'-Trimethylangelicin as a Possible Treatment for Cystic Fibrosis

自乳化制剂可提高4,6,4'-三甲基白芷素的口服生物利用度,作为囊性纤维化的潜在治疗方法

Franceschinis, Erica; Roverso, Marco; Gabbia, Daniela; De Martin, Sara; Brusegan, Matteo; Vaccarin, Christian; Bogialli, Sara; Chilin, Adriana

Improved Trimethylangelicin Analogs for Cystic Fibrosis: Design, Synthesis and Preliminary Screening

用于治疗囊性纤维化的改良型三甲基白芷素类似物:设计、合成和初步筛选

Vaccarin, Christian; Gabbia, Daniela; Franceschinis, Erica; De Martin, Sara; Roverso, Marco; Bogialli, Sara; Sacchetti, Gianni; Tupini, Chiara; Lampronti, Ilaria; Gambari, Roberto; Cabrini, Giulio; Dechecchi, Maria Cristina; Tamanini, Anna; Marzaro, Giovanni; Chilin, Adriana

Grapiprant or carprofen following ovariohysterectomy in the cat: analgesic efficacy, hematological, biochemical and urinalysis evaluation

猫卵巢子宫切除术后使用格拉匹仑或卡洛芬的镇痛效果、血液学、生化和尿液分析评价

Teixeira, Luciana G; Vaccarin, Charline V; Schimites, Paula I; Gasparotto, Jean C; Costa, Gabriela P; Griesang, Julia M; Vargas, Daniel; Bortolotto, Emanuelle D; Soares, Ana Bu; Camargo, Jéssica F; Andrade, Cínthia M; Soares, André V; Contesini, Emerson A