日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Selective disruption of RORγt-CBFβ interaction by IMU-935 prevents RORγt-dependent Th17 autoimmunity but not thymocyte development

IMU-935选择性地破坏RORγt-CBFβ相互作用可阻止RORγt依赖的Th17自身免疫,但不影响胸腺细胞发育。

Wu, Hongmin; Zhong, Xiancai; Ma, Ning; He, Zhiheng; Wang, Guanpeng; Lu, Geming; Yuan, Yate-Ching; Zhang, Wencan; Shi, Yun; Vaidehi, Nagarajan; Peelen, Evelyn; Wulff, Tanja; Gege, Christian; Kohlhof, Hella; Vitt, Daniel; Gwack, Yousang; Taniuchi, Ichiro; Xue, Hai-Hui; Sun, Zuoming

Dynamic feedback control of oncogenic tyrosine kinase signaling in acute leukemia.

急性白血病中致癌酪氨酸激酶信号的动态反馈控制。

Lee Jaewoong, Sun Ruifeng, Kume Kohei, Robinson Mark E, Cheng Zhangliang, Cosgun Kadriye Nehir, Ma Ning, Hurtz Christian, Geng Huimin, Luger Selina M, Litzow Mark R, Paietta Elisabeth, Chen Jianjun, Vaidehi Nagarajan, Müschen Markus

Stabilization versus flexibility: Detergent-dependent trade-offs in neurotensin receptor 1 GPCR ensembles

稳定性与灵活性:去垢剂依赖的神经降压素受体 1 GPCR 集合的权衡

Bower, James B; van der Velden, Wijnand J C; Gomez, Karen P; Pan, Mingzhe; Bumbak, Fabian; Vaidehi, Nagarajan; Ziarek, Joshua J

Allostery between Distant Structural Regions Dictates Selectivity in GPCR:G Protein Coupling

远端结构区域间的变构作用决定了GPCR:G蛋白偶联的选择性

Mukhaleva, Elizaveta; Sánchez Rivas, Edgardo J; Branciamore, Sergio; Rodin, Andrei S; Sivaramakrishnan, Sivaraj; Vaidehi, Nagarajan

Screening for novel chemical scaffolds targeting PCNA identifies the Hsp90alpha inhibitor SNX-2112

针对 PCNA 的新型化学骨架筛选鉴定出 Hsp90α 抑制剂 SNX-2112

Jossart, Jennifer; Ma, Ning; Haratipour, Pouya; Li, Caroline M; Jang, Christopher; Gu, Long; O'Brien, Terrence E; Vaidehi, Nagarajan; Malkas, Linda H; Hickey, Robert J; Perry, J Jefferson P

Conserved Residues in the Gα interface show subtype specificity in Gβγ coupling

Gα界面上的保守残基在Gβγ偶联中表现出亚型特异性。

Wei, Wenyuan; Taylor, H Dalton; Ma, Ning; Rodin, Andrei S; Branciamore, Sergio; Dohlman, Henrik G; Vaidehi, Nagarajan

Mapping the Ligand-dependent Remodeling of the Conformational Entropy Landscape in Neurotensin Receptor 1 by NMR-guided Molecular Simulations

利用核磁共振引导的分子模拟绘制神经降压素受体1中配体依赖性构象熵景观重塑图谱

Robson, Scott A; Bumbak, Fabian; Bhattacharya, Supriyo; van der Velden, Wijnand J C; Vaidehi, Nagarajan; Ziarek, Joshua J

Temporally resolved and interpretable machine learning model of GPCR conformational transition

具有时间分辨性和可解释性的GPCR构象转变机器学习模型

Manookian, Babgen; Mukhaleva, Elizaveta; Gogoshin, Grigoriy; Bhattacharya, Supriyo; Sivaramakrishnan, Sivaraj; Vaidehi, Nagarajan; Rodin, Andrei S; Branciamore, Sergio

Frustration in the protein-protein interface plays a central role in the cooperativity of PROTAC ternary complexes

蛋白质-蛋白质界面处的相互作用受阻在PROTAC三元复合物的协同作用中起着核心作用。

Ma, Ning; Bhattacharya, Supriyo; Muk, Sanychen; Jandova, Zuzana; Schmalhorst, Philipp S; Ghosh, Soumadwip; Le, Keith; Diers, Emelyne; Trainor, Nicole; Farnaby, William; Roy, Michael J; Kofink, Christiane; Greb, Peter; Weinstabl, Harald; Ciulli, Alessio; Bader, Gerd; Sankar, Kyra; Bergner, Andreas; Vaidehi, Nagarajan

Allosteric communication mechanism in the glucagon receptor

胰高血糖素受体中的变构通讯机制

van der Velden, Wijnand J C; Mukhaleva, Elizaveta; Vaidehi, Nagarajan