Development of cell-active BRD4-D1 selective inhibitors to decode the role of BET proteins in LPS-mediated liver inflammation
开发具有细胞活性的BRD4-D1选择性抑制剂,以揭示BET蛋白在LPS介导的肝脏炎症中的作用
期刊:European Journal of Medicinal Chemistry
影响因子:5.9
doi:10.1016/j.ejmech.2025.118519
Scholtz, Cole R; Doskey, Luke C; Kandanur, Sai Giridhar Sarma; Vail, Nora R; Roderick, Erika R; Peterson, Elliott J; Hoell, Zachariah J; Shi, Ke; Aihara, Hideki; Kostallari, Enis; Shah, Vijay H; Malhi, Harmeet; Pomerantz, William C K