日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inhibiting peptidylarginine deiminases (PAD1-4) by targeting a Ca(2+) dependent allosteric binding site.

通过靶向 Ca(2+) 依赖性变构结合位点来抑制肽基精氨酸脱亚胺酶 (PAD1-4)

Dakin Leslie A, Xing Li, Hall Justin, Ding Weidong, Vajdos Felix F, Pelker Jeffrey W, Ramsey Simeon, Balbo Paul, Sahasrabudhe Parag V, Banker Mary Ellen, Choi Won Young, Wright Stephen W, Chang Jeanne S, Curto John M, Davoren Jennifer E, Drozda Susan E, Fennell Kimberly F, Futatsugi Kentaro, Kortum Steve, Lee Katherine L, Liu Shenping, Lovering Frank, Nicki Jennifer A, Trujillo John I, Vincent Fabien, Schnute Mark E

Macrocyclic Retinoic Acid Receptor-Related Orphan Receptor C2 Inverse Agonists

大环维甲酸受体相关孤儿受体C2反向激动剂

Schnute, Mark E; Trujillo, John I; Lee, Katherine L; Unwalla, Ray; Vajdos, Felix F; Kauppi, Björn; Nuhant, Philippe; Flick, Andrew C; Crouse, Kimberly K; Zhao, Yajuan; Samuel, Amanda; Lombardo, Vincent; Taylor, Alexandria P; Brault, Amy L; Knafels, John D; Vazquez, Michael L; Berstein, Gabriel

Demonstration of In Vitro to In Vivo Translation of a TYK2 Inhibitor That Shows Cross Species Potency Differences

TYK2 抑制剂的体外至体内转化演示,显示跨物种效力差异

Brian S Gerstenberger, Mary Ellen Banker, James D Clark, Martin E Dowty, Andrew Fensome, Roger Gifford, Matthew C Griffor, Martin Hegen, Brett D Hollingshead, John D Knafels, Tsung H Lin, James F Smith, Felix F Vajdos

Aminomethyl-Derived Beta Secretase (BACE1) Inhibitors: Engaging Gly230 without an Anilide Functionality

氨甲基衍生的β-分泌酶(BACE1)抑制剂:无需苯胺官能团即可与Gly230结合

Butler, Christopher R; Ogilvie, Kevin; Martinez-Alsina, Luis; Barreiro, Gabriela; Beck, Elizabeth M; Nolan, Charles E; Atchison, Kevin; Benvenuti, Eric; Buzon, Leanne; Doran, Shawn; Gonzales, Cathleen; Helal, Christopher J; Hou, Xinjun; Hsu, Mei-Hui; Johnson, Eric F; Lapham, Kimberly; Lanyon, Lorraine; Parris, Kevin; O'Neill, Brian T; Riddell, David; Robshaw, Ashley; Vajdos, Felix; Brodney, Michael A

Suppressor of fused regulates Gli activity through a dual binding mechanism

融合抑制因子通过双重结合机制调节 Gli 活性

Merchant, Mark; Vajdos, Felix F; Ultsch, Mark; Maun, Henry R; Wendt, Ulrich; Cannon, Jennifer; Desmarais, William; Lazarus, Robert A; de Vos, Abraham M; de Sauvage, Frederic J

How to measure and predict the molar absorption coefficient of a protein

如何测量和预测蛋白质的摩尔吸光系数

Pace, C N; Vajdos, F; Fee, L; Grimsley, G; Gray, T