日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

OICR-41103 as a chemical probe for the DCAF1 WD40 domain.

OICR-41103 作为 DCAF1 WD40 结构域的化学探针

Kimani Serah W, Noureldin Mahmoud, Wilson Brian, Hoffer Laurent, Green Stuart R, Szewczyk Magdalena M, González-Álvarez Héctor, Mohammed Mohammed, Chan Manuel, Krausser Chiara, Li Alice Shi Ming, Hajian Taraneh, Tucker Sarah, Joshi Dhananjay, Saraon Punit, Thériault Brigitte, Kim Ji Sup, Santhakumar Vijayaratnam, Loppnau Peter, Li Yanjun, Seitova Almagul, Dong Aiping, Kiyota Taira, Hammann Tobias, Gehrtz Paul, Patel Bhashant, Rathod Vaibhavi, Vala Anand, Rout Bhimsen, Jagodra Paras, Brown Peter J, Aman Ahmed, Ramnauth Jailall, Poda Gennady, Uehling David, Arrowsmith Cheryl H, Barsyte-Lovejoy Dalia, Marcellus Richard, Ackloo Suzanne, Mamai Ahmed, Al-Awar Rima, Halabelian Levon

Enantioselective Chemical Probe for Chikungunya nsP2 Helicase with Antialphaviral Activity

具有抗甲病毒活性的基孔肯雅病毒nsP2解旋酶对映选择性化学探针

Muthu Ramalingam, Bose; Oh, Hans J; Sears, John D; Chen, Chun-Hsing; Vala, Anand; Liu, Shubin; Talbot, Kacey M; Hossain, Mohammed Anwar; Brown, Peter J; Houliston, Scott; Garcia Perez, Julia; Li, Fengling; Amare, Meareg G; Halfmann, Peter; Smith, Jessica L; Hirsch, Alec J; Arrowsmith, Cheryl H; Halabelian, Levon; Vargason, Ava; Couñago, Rafael M; Arnold, Jamie J; Cameron, Craig E; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M

Structure Activity of β-Amidomethyl Vinyl Sulfones as Covalent Inhibitors of Chikungunya nsP2 Cysteine Protease with Antialphavirus Activity

β-酰胺甲基乙烯基砜作为基孔肯雅病毒nsP2半胱氨酸蛋白酶共价抑制剂的结构活性及其抗甲病毒活性

Ghoshal, Anirban; Asressu, Kesatebrhan Haile; Hossain, Mohammad Anwar; Brown, Peter J; Nandakumar, Meganathan; Vala, Anand; Merten, Eric M; Sears, John D; Law, Isabella; Burdick, Jane E; Morales, Noah L; Perveen, Sumera; Pearce, Kenneth H; Popov, Konstantin I; Moorman, Nathaniel J; Heise, Mark T; Willson, Timothy M