日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Tunable Aromatic Sulfoxides and Sulfones as Cysteine-Targeting Warheads: Exploring the Structure-Reactivity Relationship

可调控的芳香族亚砜和砜作为半胱氨酸靶向弹头:探索结构-反应性关系

Nyström, Hampus; Valaka, Anna P; Kalesse, Hanna A; Håversen, Liliana; Olsson, Thomas; Gunnarsson, Anders; Schweikart, Fritz; Borén, Jan; Grøtli, Morten

Potent Fluorescent Probe for Target-Engagement Studies of Allosteric Pyruvate Kinase Modulators

用于变构丙酮酸激酶调节剂靶点结合研究的高效荧光探针

Nilsson, Oscar; Valaka, Anna P; Håversen, Liliana; Bogucka, Agnieszka; Köteles, István; Brear, Paul; Rutberg, Mikael; Gunnarsson, Anders; Hyvönen, Marko; Grøtli, Morten

Design and application of a fluorescent probe for imaging of endogenous Bruton's tyrosine kinase with preserved enzymatic activity

设计并应用一种荧光探针,用于成像内源性布鲁顿酪氨酸激酶,该探针保留了酶活性。

Valaka, Anna P; Nyström, Hampus; Håversen, Liliana; Benitez-Martin, Carlos; Schäfer, Clara; Jang, Woo Suk; Camponeschi, Alessandro; Andréasson, Joakim; Borén, Jan; Grøtli, Morten