日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A synergistic interaction between PRMT5 and LSD1 inhibitors in AML.

PRMT5 和 LSD1 抑制剂在急性髓系白血病中存在协同作用。

Param Nesteene Joy, Arceci Elisa, Fiorentino Francesco, Pignata Luca, Torre Denis, Gutiérrez-Trejo Nayeli, Fong Jia Yi, Goy Pierre-Alexis, Han Brenda Y, Lambona Chiara, Di Bello Elisabetta, Castiello Carola, Barone Marco, Schwarz Megan, Arrowsmith Cheryl, Ito Koichi, Scherle Peggy, Wee Dave Keng Boon, Ndoye Steven, Tabaglio Tommaso, Jeyasekharan Anand D, Lakshmanan Manikandan, Cirilli Roberto, Habisch Hansjörg, Madl Tobias, Mattevi Andrea, Valente Sergio, Mai Antonello, Guccione Ernesto

Dynamic epigenetic regulation of BCLAF1 splicing in acute myeloid leukemia

急性髓系白血病中BCLAF1剪接的动态表观遗传调控

Sgueglia, Giulia; Massaro, Crescenzo; Muro, Annamaria; Lettiero, Ida; D'Agostino, Erika; Favale, Gregorio; Simonelli, Nicla; Del Gaudio, Nunzio; Carafa, Vincenzo; De Marchi, Tommaso; Rotili, Dante; Valente, Sergio; Mai, Antonello; Sbardella, Gianluca; De Simone, Mariacarla; Altucci, Lucia; Dell'Aversana, Carmela

Combined computational and classical medicinal chemistry procedure to disclose novel pyrrole-based compounds as potential antituberculosis agents

结合计算和经典药物化学方法,发现新型吡咯类化合物作为潜在的抗结核药物。

Ragno, Rino; Zwergel, Clemens; Valente, Sergio; Astolfi, Roberta; Lambona, Chiara; Proia, Eleonora; Giuliani, Lidia; Franzblau, Scott G; Fioravanti, Rossella; Mai, Antonello

Long noncoding RNA H19 promotes the acquisition of a mesenchymal-like invasive phenotype in mesothelial primary cells through an HDAC1-mediated WT1/Sp1 switch.

长链非编码 RNA H19 通过 HDAC1 介导的 WT1/Sp1 转换促进间皮原代细胞获得间充质样侵袭表型

Bontempi Giulio, Michetti Federica, Terri Michela, Battistelli Cecilia, Conigliaro Alice, Garbo Sabrina, Montaldo Claudia, Valente Sergio, Zwergel Clemens, Mai Antonello, Nahavandi Araghi Azadeh, Domenici Alessandro, Menè Paolo, Tripodi Marco, Strippoli Raffaele

Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells

发现具有抗癌细胞增殖活性的首创碳酸酐酶/组蛋白去乙酰化酶双重抑制剂

Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T

Advancements in Hydrazide-Based HDAC Inhibitors: A Review of Recent Developments and Therapeutic Potential

基于酰肼的HDAC抑制剂的研究进展:近期进展及治疗潜力综述

Raucci, Alessia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello

Quinoline-Based DNA Methyltransferase Inhibitors Featuring Basic Side Chains: Design, Synthesis, and Insight in Biochemical and Anticancer Cell Properties

具有碱性侧链的喹啉类DNA甲基转移酶抑制剂:设计、合成及其生化和抗癌细胞特性研究

Zwergel, Clemens; Lambona, Chiara; Fioravanti, Rossella; Raucci, Alessia; Fiorentino, Francesco; Nchugoua Tchieh, Guilaine; Jallet, Corinne; Lacroix, Laurent; Pierrettori, Michela; Pellegrini, Francesca Romana; Xiong, Yan; Jin, Jian; Arimondo, Paola; Trisciuoglio, Daniela; Mai, Antonello; Valente, Sergio

Cardioprotection Through Pharmacological Activation of Sirtuin 5 in a Murine Model of Acute Myocardial Infarction

在急性心肌梗死小鼠模型中,通过药物激活Sirtuin 5发挥心脏保护作用

Castiello, Carola; Efentakis, Panagiotis; Nikolaou, Panagiota-Efstathia; Symeonidi, Lydia; Chania, Christina; Barla, Ioanna; Akrani, Ifigeneia; Kostomitsopoulos, Nikolaos; Gikas, Evangelos; Thomaidis, Nikolaos S; Mikros, Emmanuel; Kleinbongard, Petra; Fioravanti, Rossella; Zwergel, Clemens; Valente, Sergio; Mai, Antonello; Andreadou, Ioanna

A Combined SIRT5 Activation and SIRT3 Inhibition Prevents Breast Cancer Spheroids Growth by Reducing HIF-1α and Mitophagy

SIRT5激活和SIRT3抑制联合作用可通过减少HIF-1α和线粒体自噬来阻止乳腺癌球体的生长

Barreca, Federica; Aventaggiato, Michele; Cristina, Mario; Sansone, Luigi; Belli, Manuel; Lista, Maria Beatrice; Francisci, Gaia; Valente, Sergio; Rotili, Dante; Mai, Antonello; Russo, Matteo Antonio; Tafani, Marco

Optimization of Transcription Factor-Driven Neuronal Differentiation from Human Induced Pluripotent Stem Cells for Disease Modelling and Drug Screening

利用转录因子驱动的人类诱导多能干细胞神经元分化优化方法构建疾病模型和药物筛选

Martina Servetti ,Martino Caramia ,Giulia Parodi ,Fabrizio Loiacono ,Ennio Nano ,Giorgia Biddau ,Lorenzo Ferrando ,Lisastella Morinelli ,Pierluigi Valente ,Sergio Martinoia ,Andrea Escelsior ,Gianluca Serafini ,Serena Tamburro ,Simona Baldassari ,Anna Fassio ,Fabio Benfenati ,Anna Corradi # ,Bruno Sterlini #