日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CACHE Challenge #3: Targeting the Nsp3 Macrodomain of SARS-CoV-2

CACHE挑战赛#3:靶向SARS-CoV-2的Nsp3宏结构域

Herasymenko, Oleksandra; Silva, Madhushika; Correy, Galen J; Abu-Saleh, Abd Al-Aziz A; Ackloo, Suzanne; Arrowsmith, Cheryl; Ashworth, Alan; Ban, Fuqiang; Beck, Hartmut; Bishop, Kevin P; Bohórquez, Hugo J; Bolotokova, Albina; Breznik, Marko; Chau, Irene; Chen, Yu; Cherkasov, Artem; Dehaen, Wim; Della Corte, Dennis; Denzinger, Katrin; Doering, Niklas P; Edfeldt, Kristina; Edwards, Aled; Fayne, Darren; Gentile, Francesco; Gibson, Elisa; Gokdemir, Ozan; Gunnarsson, Anders; Günther, Judith; Irwin, John J; Jensen, Jan Halborg; Harding, Rachel J; Hillisch, Alexander; Hoffer, Laurent; Hogner, Anders; Hutchinson, Ashley; Kandwal, Shubhangi; Karlova, Andrea; Koirala, Kushal; Kotelnikov, Sergei; Kozakov, Dima; Lee, Juyong; Lee, Soowon; Lessel, Uta; Liu, Sijie; Liu, Xuefeng; Loppnau, Peter; Meiler, Jens; Moretti, Rocco; Moroz, Yurii S; Muvva, Charuvaka; Oprea, Tudor I; Paige, Brooks; Pandit, Amit; Park, Keunwan; Poda, Gennady; Protopopov, Mykola V; Pütter, Vera; Ravichandran, Rahul; Rognan, Didier; Rosta, Edina; Sabnis, Yogesh; Scott, Thomas; Seitova, Almagul; Sharma, Purshotam; Sindt, François; Song, Minghu; Steinmann, Casper; Stevens, Rick; Talagayev, Valerij; Tararina, Valentyna V; Tarkhanova, Olga; Tingey, Damon; Trant, John F; Treleaven, Dakota; Tropsha, Alexander; Walters, Patrick; Wells, Jude; Westermaier, Yvonne; Wolber, Gerhard; Wortmann, Lars; Zheng, Shuangjia; Fraser, James S; Schapira, Matthieu

Exercise and Sports Among Working-Age Citizens in Lithuania Since the COVID-19 Pandemic: An Annual Comparative Study (2021-2024)

新冠疫情以来立陶宛劳动年龄公民的运动与体育活动:年度比较研究(2021-2024)

Arlauskas, Rokas; Austys, Donatas; Stukas, Rimantas; Dobrovolskij, Valerij; Rimkevičius, Arūnas; Bulotaitė, Gabija

Primary sclerosing cholangitis in children: a single-center experience and evaluation of prognostic markers

儿童原发性硬化性胆管炎:单中心经验及预后标志物评估

Vlckova, Eva; Hradsky, Ondrej; Semjonov, Valerij; Durilova, Marianna; Kazeka, Denis; Kubat, Michal; Lerchova, Tereza; Bronsky, Jiri; Mitrova, Katarina

Discovery of Novel Isoxazole-Based Small-Molecule Toll-Like Receptor 8 Antagonists

发现新型异噁唑类小分子 Toll 样受体 8 拮抗剂

Matziol, Troy; Talagayev, Valerij; Slokan, Tjaša; Strašek Benedik, Nika; Holze, Janine; Sova, Matej; Wolber, Gerhard; Weindl, Günther

RASER for Increased Spectral Resolution in Carbon-13 NMR

RASER技术可提高碳-13核磁共振谱的分辨率

Nelson, Christopher; Schmidt, Andreas B; Adelabu, Isaiah; Nantogma, Shiraz; Dilday, Seth; Volya, Nicholas; Mandzhieva, Iuliia; Kiselev, Valerij G; Abdurraheem, Abubakar; de Maissin, Henri; Lehmkuhl, Sören; Appelt, Stephan; Chekmenev, Eduard Y; Theis, Thomas

Structure-based virtual screening identifies potent CD28 inhibitors that suppress T cell co-stimulation in cellular and mucosal models.

基于结构的虚拟筛选鉴定出有效的 CD28 抑制剂,这些抑制剂能够抑制细胞和粘膜模型中的 T 细胞共刺激。

Upadhyay Saurabh, Talagayev Valerij, Cho Sungwoo, Wolber Gerhard, Gabr Moustafa

Agonists and Antagonists Show Different Unbinding Paths from the TLR8 Receptor

激动剂和拮抗剂从TLR8受体上解离的途径不同

Talagayev, Valerij; Wolber, Gerhard; Nunes-Alves, Ariane

OpenMMDL - Simplifying the Complex: Building, Simulating, and Analyzing Protein-Ligand Systems in OpenMM

OpenMMDL——化繁为简:在OpenMM中构建、模拟和分析蛋白质-配体系统

Talagayev, Valerij; Chen, Yu; Doering, Niklas Piet; Obendorf, Leon; Denzinger, Katrin; Puls, Kristina; Lam, Kevin; Liu, Sijie; Wolf, Clemens Alexander; Noonan, Theresa; Breznik, Marko; Knaus, Petra; Wolber, Gerhard

CACHE Challenge #2: Targeting the RNA Site of the SARS-CoV-2 Helicase Nsp13

CACHE挑战#2:靶向SARS-CoV-2解旋酶Nsp13的RNA位点

Herasymenko, Oleksandra; Silva, Madhushika; Abu-Saleh, Abd Al-Aziz A; Ahmad, Ayaz; Alvarado-Huayhuaz, Jesus; Arce, Oscar E A; Armstrong, Roly J; Arrowsmith, Cheryl; Bachta, Kelly E; Beck, Hartmut; Berta, Denes; Bieniek, Mateusz K; Blay, Vincent; Bolotokova, Albina; Bourne, Philip E; Breznik, Marko; Brown, Peter J; Campbell, Aaron D G; Carosati, Emanuele; Chau, Irene; Cole, Daniel J; Cree, Ben; Dehaen, Wim; Denzinger, Katrin; Dos Santos Machado, Karina; Dunn, Ian; Durai, Prasannavenkatesh; Edfeldt, Kristina; Edwards, Aled; Fayne, Darren; Felfoldi, Daniel; Friston, Kallie; Ghiabi, Pegah; Gibson, Elisa; Günther, Judith; Gunnarsson, Anders; Hillisch, Alexander; Houston, Douglas R; Jensen, Jan Halborg; Harding, Rachel J; Harris, Kate S; Hoffer, Laurent; Hogner, Anders; Horton, Joshua T; Houliston, Scott; Hultquist, Judd F; Hutchinson, Ashley; Irwin, John J; Jukič, Marko; Kandwal, Shubhangi; Karlova, Andrea; Katis, Vittorio L; Kich, Ryan P; Kireev, Dmitri; Koes, David; Inniss, Nicole L; Lessel, Uta; Liu, Sijie; Loppnau, Peter; Lu, Wei; Martino, Sam; McGibbon, Miles; Meiler, Jens; Mettu, Akhila; Money-Kyrle, Sam; Moretti, Rocco; Moroz, Yurii S; Muvva, Charuvaka; Newman, Joseph A; Obendorf, Leon; Paige, Brooks; Pandit, Amit; Park, Keunwan; Perveen, Sumera; Pirie, Rachael; Poda, Gennady; Protopopov, Mykola; Pütter, Vera; Ricci, Federico; Roper, Natalie J; Rosta, Edina; Rzhetskaya, Margarita; Sabnis, Yogesh; Satchell, Karla J F; Schmitt Kremer, Frederico; Scott, Thomas; Seitova, Almagul; Steinmann, Casper; Talagayev, Valerij; Tarkhanova, Olga O; Tatum, Natalie J; Treleaven, Dakota; Velasque Werhli, Adriano; Walters, W Patrick; Wang, Xiaowen; Wells, Jude; Wells, Geoffrey; Westermaier, Yvonne; Wolber, Gerhard; Wortmann, Lars; Zhang, Jixian; Zhao, Zheng; Zheng, Shuangjia; Schapira, Matthieu

An Ongoing Search for Multitarget Ligands as Potential Agents for Diabetes Mellitus and Its Long-Term Complications: New Insights into (5-Arylidene-4-oxothiazolidin-3-yl)alkanoic Acid Derivatives

持续探索多靶点配体作为糖尿病及其长期并发症的潜在治疗药物:对(5-亚芳基-4-氧代噻唑烷-3-基)烷酸衍生物的新认识

Maccari, Rosanna; Ottanà, Rosaria; Talagayev, Valerij; Moschini, Roberta; Balestri, Francesco; Felice, Francesca; Iannuccilli, Francesca; Sardelli, Gemma; Sodano, Rebecca; Wolber, Gerhard; Paoli, Paolo; Del Corso, Antonella