日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Partitioning of the initial catalytic steps of leucyl-tRNA synthetase is driven by an active site peptide-plane flip

亮氨酰-tRNA合成酶初始催化步骤的划分是由活性位点肽平面翻转驱动的。

Pang, Luping; Zanki, Vladimir; Strelkov, Sergei V; Van Aerschot, Arthur; Gruic-Sovulj, Ita; Weeks, Stephen D

Discovery of novel druggable pockets on polyomavirus VP1 through crystallographic fragment-based screening to develop capsid assembly inhibitors

通过基于晶体学片段的筛选发现多瘤病毒VP1上的新型可成药口袋,以开发衣壳组装抑制剂

Osipov, Evgenii M; Munawar, Ali H; Beelen, Steven; Fearon, Daren; Douangamath, Alice; Wild, Conor; Weeks, Stephen D; Van Aerschot, Arthur; von Delft, Frank; Strelkov, Sergei V

Synthetic strategy and antiviral evaluation of diamide containing heterocycles targeting dengue and yellow fever virus

合成策略及含二酰胺杂环化合物对登革热病毒和黄热病毒的抗病毒活性评价

Saudi, Milind; Zmurko, Joanna; Kaptein, Suzanne; Rozenski, Jef; Gadakh, Bharat; Chaltin, Patrick; Marchand, Arnaud; Neyts, Johan; Van Aerschot, Arthur

The RimL transacetylase provides resistance to translation inhibitor microcin C

RimL转乙酰酶赋予其对翻译抑制剂微生素C的抗性。

Kazakov, Teymur; Kuznedelov, Konstantin; Semenova, Ekaterina; Mukhamedyarov, Damir; Datsenko, Kirill A; Metlitskaya, Anastasija; Vondenhoff, Gaston H; Tikhonov, Anton; Agarwal, Vinayak; Nair, Satish; Van Aerschot, Arthur; Severinov, Konstantin

Structural and functional characterization of microcin C resistance peptidase MccF from Bacillus anthracis.

炭疽杆菌微生素 C 抗性肽酶 MccF 的结构和功能表征

Nocek Boguslaw, Tikhonov Anton, Babnigg Gyorgy, Gu Minyi, Zhou Min, Makarova Kira S, Vondenhoff Gaston, Van Aerschot Arthur, Kwon Keehwan, Anderson Wayne F, Severinov Konstantin, Joachimiak Andrzej

Crystallization and preliminary X-ray study of the D-altritol oligonucleotide GTGTACAC.

D-altritol 寡核苷酸 GTGTACAC 的结晶和初步 X 射线研究

Ovaere Margriet, Van Aerschot Arthur, Abramov Mikhail, Herdewijn Piet, Van Meervelt Luc

A large-scale chemical modification screen identifies design rules to generate siRNAs with high activity, high stability and low toxicity

大规模化学修饰筛选确定了生成具有高活性、高稳定性和低毒性的siRNA的设计规则。

Bramsen, Jesper B; Laursen, Maria B; Nielsen, Anne F; Hansen, Thomas B; Bus, Claus; Langkjaer, Niels; Babu, B Ravindra; Højland, Torben; Abramov, Mikhail; Van Aerschot, Arthur; Odadzic, Dalibor; Smicius, Romualdas; Haas, Jens; Andree, Cordula; Barman, Jharna; Wenska, Malgorzata; Srivastava, Puneet; Zhou, Chuanzheng; Honcharenko, Dmytro; Hess, Simone; Müller, Elke; Bobkov, Georgii V; Mikhailov, Sergey N; Fava, Eugenio; Meyer, Thomas F; Chattopadhyaya, Jyoti; Zerial, Marino; Engels, Joachim W; Herdewijn, Piet; Wengel, Jesper; Kjems, Jørgen

Inhibition of MDR1 gene expression by chimeric HNA antisense oligonucleotides

嵌合HNA反义寡核苷酸对MDR1基因表达的抑制作用

Kang, Hyunmin; Fisher, Michael H; Xu, Dong; Miyamoto, Yuko J; Marchand, Arnaud; Van Aerschot, Arthur; Herdewijn, Piet; Juliano, Rudolph L

Chemical incorporation of 1-methyladenosine into oligonucleotides

将1-甲基腺苷化学掺入寡核苷酸中

Mikhailov, Sergey N; Rozenski, Jef; Efimtseva, Ekaterina V; Busson, Roger; Van Aerschot, Arthur; Herdewijn, Piet