日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacological tools to modulate ordered membrane domains and order-dependent protein function

利用药理学工具调节有序膜结构域和有序依赖性蛋白质功能

Stefanski, Katherine M; Huang, Hui; Luu, Dustin D; Li, Geoffrey C; Hutchison, James M; Saksena, Nilabh; Fisch, Alexander J; Hasaka, Thomas P; Bauer, Joshua A; Kenworthy, Anne K; Van Horn, Wade D; Sanders, Charles R

TRPM8 Protein Dynamics Correlates with Ligand Structure and Cellular Function.

TRPM8 蛋白动力学与配体结构和细胞功能相关

Mebrat Mubark D, Luu Dustin D, Hilton Jacob K, Kim Minjoo, Parrott Kaitlyn, Cherry Brian R, Levitus Marcia, Journigan V Blair, Van Horn Wade D

Detection of non-native species formed during fibrillization of the myocilin olfactomedin domain

检测肌纤蛋白嗅觉介素结构域纤维化过程中形成的非天然物种

Scelsi, Hailee F; Close, Emily G S; Huard, Dustin J E; Dunn, Elijah; Bogdanović, Nebojša; Mudiyanselage, Sonali H W; Grant, Arshay; Stagg, Scott M; Schmidt-Krey, Ingeborg; Van Horn, Wade D; Lieberman, Raquel L

Veraguamide E, a Marine Cyanobacterial Depsipeptide Targeting σ(2)R/TMEM97: Chemical and Neurobiological Characterization

Veraguamide E,一种靶向 σ(2)R/TMEM97 的海洋蓝藻缩肽:化学和神经生物学表征

Sotelo-Morales, Jesus E; Mofidi Tabatabaei, Sahar; Fofie, Christian K; Fosu, Kelvin K; Dodd-O, Joseph B; Simcik, Rebekah D; Tack, See H; Soto-Reyes, Miguel J; Yousuf, Muhammad Saad; Caro-Diaz, Eduardo J E; Kumar, Vivek A; Van Horn, Wade D; Kolber, Benedict; Tidgewell, Kevin J

Pharmacological Tools to Modulate Ordered Membrane Domains and Order-Dependent Protein Function

利用药理学工具调节有序膜结构域和有序依赖性蛋白质功能

Stefanski, Katherine M; Huang, Hui; Luu, Dustin D; Hutchison, James M; Saksena, Nilabh; Fisch, Alexander J; Hasaka, Thomas P; Bauer, Joshua A; Kenworthy, Anne K; Van Horn, Wade D; Sanders, Charles R

TRPM8 protein dynamics correlates with ligand structure and cellular function.

TRPM8 蛋白动力学与配体结构和细胞功能相关

Mebrat Mubark D, Luu Dustin D, Hilton Jacob K, Kim Minjoo, Parrott Kaitlyn, Cherry Brian R, Levitus Marcia, Journigan V Blair, Van Horn Wade D

Uracil-DNA glycosylase efficiency is modulated by substrate rigidity

尿嘧啶-DNA糖苷酶的效率受底物刚性的调节

Orndorff, Paul B; Poddar, Souvik; Owens, Aerial M; Kumari, Nikita; Ugaz, Bryan T; Amin, Samrat; Van Horn, Wade D; van der Vaart, Arjan; Levitus, Marcia

A molecular perspective on identifying TRPV1 thermosensitive regions and disentangling polymodal activation

从分子层面识别TRPV1热敏区域并解析其多模态激活机制

Luu, Dustin D; Owens, Aerial M; Mebrat, Mubark D; Van Horn, Wade D

CryoFold: determining protein structures and data-guided ensembles from cryo-EM density maps

CryoFold:利用冷冻电镜密度图确定蛋白质结构和数据引导的集合

Shekhar, Mrinal; Terashi, Genki; Gupta, Chitrak; Sarkar, Daipayan; Debussche, Gaspard; Sisco, Nicholas J; Nguyen, Jonathan; Mondal, Arup; Vant, John; Fromme, Petra; Van Horn, Wade D; Tajkhorshid, Emad; Kihara, Daisuke; Dill, Ken; Perez, Alberto; Singharoy, Abhishek

Structural and in Vitro Functional Characterization of a Menthyl TRPM8 Antagonist Indicates Species-Dependent Regulation

薄荷基TRPM8拮抗剂的结构和体外功能表征表明其调控存在物种依赖性。

Journigan, V Blair; Alarcón-Alarcón, David; Feng, Zhiwei; Wang, Yuanqiang; Liang, Tianjian; Dawley, Denise C; Amin, A R M Ruhul; Montano, Camila; Van Horn, Wade D; Xie, Xiang-Qun; Ferrer-Montiel, Antonio; Fernández-Carvajal, Asia