日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Characterization of Novel Sigma Receptor Ligands Derived from Multicomponent Reactions as Efficacious Treatments for Neuropathic Pain

表征源自多组分反应的新型σ受体配体作为治疗神经性疼痛的有效方法

Shinouchi, Ryosuke; Turgutalp, Bengisu; Ople, Rohini S; Eans, Shainnel O; Williams, Ashai K; Hammond, Haylee R; Varadi, Andras; Dardashti, Rebecca Notis; Majumdar, Susruta; McLaughlin, Jay P

Synthesis and Pharmacology of a Morphinan-Derived Dual Mu-Kappa Opioid Receptor Agonist Analgesic.

吗啡烷衍生的双重μ-κ阿片受体激动剂镇痛药的合成与药理学研究

Varga Balazs R, Uprety Rajendra, Paul Barnali, Knoll Alexis, Ramos-Gonzalez Nokomis, Appourchaux Kevin, Taylor Tori, Turgutalp Bengisu, Shinouchi Ryosuke, Eans Shainnel O, Williams Ashai K, Vasquez-Grinnell Steven G, Zaidi Saheem, Nazarova Antonina L, Varadi Andras, Le Rouzic Valerie, Brown Taylor G, Martinez Shani, Ansonoff Michael, Dardashti Rebecca Notis, Hunkele Amanda, Subrath Joan, Welch Matthew, Xu Jin, Rossi Grace C, Pintar John, Pasternak Gavril W, Katritch Vsevolod, McLaughlin Jay P, Pan Ying Xian, Majumdar Susruta

Design, Synthesis, and Preclinical Efficacy of Novel Nonretinoid Antagonists of Retinol-Binding Protein 4 in the Mouse Model of Hepatic Steatosis

在小鼠肝脂肪变性模型中,设计、合成并评估新型非视黄醇类视黄醇结合蛋白4拮抗剂的临床前疗效

Cioffi, Christopher L; Racz, Boglarka; Varadi, Andras; Freeman, Emily E; Conlon, Michael P; Chen, Ping; Zhu, Lei; Kitchen, Douglas B; Barnes, Keith D; Martin, William H; Pearson, Paul G; Johnson, Graham; Blaner, William S; Petrukhin, Konstantin

Genetic dissociation of morphine analgesia from hyperalgesia in mice

小鼠吗啡镇痛作用与痛觉过敏的遗传分离

Marrone, Gina F; Le Rouzic, Valerie; Varadi, Andras; Xu, Jin; Rajadhyaksha, Anjali M; Majumdar, Susruta; Pan, Ying-Xian; Pasternak, Gavril W