Discovering Uncharted Binding Pockets on E3 Ligases Leads to the Identification of FBW7 Allosteric Modulators
发现E3连接酶上未知的结合口袋,从而鉴定出FBW7变构调节剂
期刊:Advanced Science
影响因子:14.1
doi:10.1002/advs.202506068
Martínez-Cartró, Míriam; Serrano-Morrás, Álvaro; Bertran-Mostazo, Andrea; Castaño-Muñiz, Roger; Scaffidi, Salvatore; Ivanova, Varbina; Csorba, Noémi; Simon, József; Ábrányi-Balogh, Péter; Li, Yunfeng; Keserü, György M; Hao, Bing; Barril, Xavier; Galdeano, Carles