日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Enzymes in secondary pharmacology screening panels: is there room for improvement?

二级药理学筛选组合中的酶:还有改进的空间吗?

Maciag, Monika; Karamyan, Vardan T

The Missing Enzymes: A Call to Update Pharmacological Profiling Practices for Better Drug Safety Assessment

缺失的酶:呼吁更新药理学分析方法,以更好地评估药物安全性

Maciag, Monika; Karamyan, Vardan T

Assessing the effects of antidepressant use on stroke recurrence and related outcomes in ischemic stroke patients: a propensity score matched analysis

评估抗抑郁药使用对缺血性卒中患者卒中复发及相关结局的影响:一项倾向评分匹配分析

Alamri, Faisal F; Almarghalani, Daniyah A; Alatawi, Yasser; Alraddadi, Eman A; Babateen, Omar; Alayyafi, Ahmed; Almalki, Ziyad; Alsalhi, Khaled; Alzahrani, Khaled; Alghamdi, Ahmed; Aldera, Hussain; Karamyan, Vardan T

Structural basis of divergent substrate recognition and inhibition of human neurolysin

人类神经溶酶体不同底物识别和抑制的结构基础

Ke Shi, Sounak Bagchi, Jordis Bickel, Shiva H Esfahani, Lulu Yin, Tiffany Cheng, Vardan T Karamyan, Hideki Aihara

In-Vivo and Ex-Vivo Brain Uptake Studies of Peptidomimetic Neurolysin Activators in Healthy and Stroke Animals

肽类神经溶酶激活剂在健康和中风动物体内和体外的脑摄取研究

Saeideh Nozohouri, Shiva Hadi Esfahani, Behnam Noorani, Dhaval Patel, Heidi Villalba, Yashwardhan Ghanwatkar, Md Shafikur Rahman, Yong Zhang, Ulrich Bickel, Paul C Trippier, Vardan T Karamyan, Thomas J Abbruscato

Estrogen Metabolite 2-Methoxyestradiol Attenuates Blood Pressure in Hypertensive Rats by Downregulating Angiotensin Type 1 Receptor

雌激素代谢物 2-甲氧基雌二醇通过下调血管紧张素 1 型受体降低高血压大鼠的血压

Yong Zhang, Benard O Ogola, Laxmi Iyer, Vardan T Karamyan, Thomas Thekkumkara

Is Diminazene an Angiotensin-Converting Enzyme 2 (ACE2) Activator? Experimental Evidence and Implications

二甲胺嗪是血管紧张素转换酶 2 (ACE2) 激活剂吗?实验证据和启示

Shiva Hadi Esfahani, Srinidhi Jayaraman, Vardan T Karamyan

Structure-activity relationship studies of functionalized aromatic peptidomimetics as neurolysin activators

功能化芳香肽模拟物作为神经溶素激活剂的构效关系研究

Rahman, Md Shafikur; Esfahani, Shiva Hadi; Nozohouri, Saeideh; Kumari, Shikha; Kocot, Joanna; Zhang, Yong; Abbruscato, Thomas J; Karamyan, Vardan T; Trippier, Paul C

Discovery of First-in-Class Peptidomimetic Neurolysin Activators Possessing Enhanced Brain Penetration and Stability

发现具有增强脑渗透性和稳定性的首创肽类神经溶酶激活剂

Md Shafikur Rahman, Shikha Kumari, Shiva Hadi Esfahani, Saeideh Nozohouri, Srinidhi Jayaraman, Nihar Kinarivala, Joanna Kocot, Andrew Baez, Delaney Farris, Thomas J Abbruscato, Vardan T Karamyan, Paul C Trippier

The role of peptidase neurolysin in neuroprotection and neural repair after stroke

肽酶神经溶素在卒中后神经保护和神经修复中的作用

Karamyan, Vardan T