Discovery of KRB-456, a KRAS G12D Switch-I/II Allosteric Pocket Binder That Inhibits the Growth of Pancreatic Cancer Patient-derived Tumors
发现 KRB-456,一种可抑制胰腺癌患者来源肿瘤生长的 KRAS G12D Switch-I/II 变构口袋结合剂
期刊:Cancer Research Communications
影响因子:2
doi:10.1158/2767-9764.CRC-23-0222
Aslamuzzaman Kazi #, Alok Ranjan #, Vasantha Kumar M V, Bogos Agianian, Martin Garcia Chavez, Vignesh Vudatha, Rui Wang, Rajanikanth Vangipurapu, Liwei Chen, Perry Kennedy, Karthikeyan Subramanian, Jonathan C K Quirke, Francisca Beato, Patrick W Underwood, Jason B Fleming, Jose Trevino, Paul J Herge