Crystal structures of DCAF1-PROTAC-WDR5 ternary complexes provide insight into DCAF1 substrate specificity
DCAF1-PROTAC-WDR5三元复合物的晶体结构揭示了DCAF1的底物特异性
期刊:Nature Communications
影响因子:14.7
doi:10.1038/s41467-024-54500-x
Mark F Mabanglo # ,Brian Wilson # ,Mahmoud Noureldin # ,Serah W Kimani ,Ahmed Mamai ,Chiara Krausser ,Héctor González-Álvarez ,Smriti Srivastava ,Mohammed Mohammed ,Laurent Hoffer ,Manuel Chan ,Jamie Avrumutsoae ,Alice Shi Ming Li ,Taraneh Hajian ,Sarah Tucker ,Stuart Green ,Magdalena Szewczyk ,Dalia Barsyte-Lovejoy ,Vijayaratnam Santhakumar ,Suzanne Ackloo ,Peter Loppnau ,Yanjun Li ,Almagul Seitova ,Taira Kiyota ,Jue George Wang ,Gilbert G Privé ,Douglas A Kuntz ,Bhashant Patel ,Vaibhavi Rathod ,Anand Vala ,Bhimsen Rout ,Ahmed Aman ,Gennady Poda ,David Uehling ,Jailall Ramnauth ,Levon Halabelian ,Richard Marcellus ,Rima Al-Awar ,Masoud Vedadi