日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Screening apelin analogues and a small molecule agonist as effective cardiovascular therapeutics against reperfusion injury

筛选apelin类似物和小分子激动剂作为对抗再灌注损伤的有效心血管治疗药物

Wijewardane, Anjalee; Fernandez, Kleinberg X; Zhang, Anran; Fischer, Conrad; Nagahawatta, Dineth P; Iturrioz, Xavier; Avet, Charlotte; Heard, Bethan L; Llorens-Cortes, Catherine; Oudit, Gavin Y; Bouvier, Michel; Vederas, John C

Structure and inhibition of diaminopimelic acid epimerase by slow-binding α-methyl amino acids

慢结合α-甲基氨基酸对二氨基庚二酸差向异构酶的结构和抑制作用

Lamer, Tess; Chen, Pu; Catenza, Karizza; Perov, Ilia; L, Bethan; Hsiao, Yu-Ting; Van Oers, Tayla J; Lemieux, M Joanne; Vederas, John C

Solution Structure of the Broad-Spectrum Bacteriocin Garvicin Q

广谱细菌素 Garvicin Q 的溶液结构

Mallett, Tyler; Lamer, Tess; Aleksandrzak-Piekarczyk, Tamara; McKay, Ryan T; Catenza, Karizza; Sit, Clarissa; Rainey, Jan K; Towle-Straub, Kaitlyn M; Vederas, John C; van Belkum, Marco J

Structural insights into the nirmatrelvir-resistant SARS-CoV-2 M(pro) L50F/E166A/L167F triple mutant-inhibitor-complex reveal strategies for next generation coronaviral inhibitor design

对耐尼马曲韦的SARS-CoV-2 M(pro) L50F/E166A/L167F三突变体-抑制剂复合物的结构解析揭示了下一代冠状病毒抑制剂的设计策略。

Fischer, Conrad; Lu, Jimmy; van Belkum, Marco J; Demmon, Sydney; Chen, Pu; Wang, Chaoxiang; Van Oers, Tayla J; Lamer, Tess; Lemieux, M Joanne; Vederas, John C

A Structural Comparison of Oral SARS-CoV-2 Drug Candidate Ibuzatrelvir Complexed with the Main Protease (M(pro)) of SARS-CoV-2 and MERS-CoV

口服SARS-CoV-2候选药物伊布扎瑞韦与SARS-CoV-2和MERS-CoV主要蛋白酶(M(pro))复合物的结构比较

Chen, Pu; Van Oers, Tayla J; Arutyunova, Elena; Fischer, Conrad; Wang, Chaoxiang; Lamer, Tess; van Belkum, Marco J; Young, Howard S; Vederas, John C; Lemieux, M Joanne

Assessment of optimized FRET substrates as universal corona- and picornavirus main protease substrates for screening assays

评估优化的FRET底物作为冠状病毒和微小核糖核酸病毒通用主蛋白酶底物在筛选试验中的应用

Fischer, Conrad; Van Oers, Tayla J; van Belkum, Marco J; Lamer, Tess; Romney, Aaron; Chen, Pu; Lemieux, M Joanne; Vederas, John C

Discovery, characterization, and structure of a cofactor-independent histidine racemase from the oral pathogen Fusobacterium nucleatum

从口腔病原体具核梭杆菌中发现、表征和解析了一种不依赖辅因子的组氨酸消旋酶的结构

Lamer, Tess; Chen, Pu; Venter, Marie J; van Belkum, Marco J; Wijewardane, Anjalee; Wu, Chenggang; Lemieux, M Joanne; Vederas, John C

Lactococcus lactis mutants resistant to lactococcin A and garvicin Q reveal missense mutations in the sugar transport domain of the mannose phosphotransferase system

对乳酸乳球菌素A和加维菌素Q具有抗性的突变体揭示了甘露糖磷酸转移酶系统糖转运结构域中的错义突变。

van Belkum, Marco J; Aleksandrzak-Piekarczyk, Tamara; Lamer, Tess; Vederas, John C

Author Correction: Genetically encoded discovery of perfluoroaryl macrocycles that bind to albumin and exhibit extended circulation in vivo

作者更正:基因编码发现的与白蛋白结合并在体内表现出延长循环时间的全氟芳基大环化合物

Wong, Jeffrey Y K; Ekanayake, Arunika I; Kharchenko, Serhii; Kirberger, Steven E; Qiu, Ryan; Kelich, Payam; Sarkar, Susmita; Li, Jiaqian; Fernandez, Kleinberg X; Alvizo-Paez, Edgar R; Miao, Jiayuan; Kalhor-Monfared, Shiva; John, J Dwyer; Kang, Hongsuk; Choi, Hwanho; Nuss, John M; Vederas, John C; Lin, Yu-Shan; Macauley, Matthew S; Vukovic, Lela; Pomerantz, William C K; Derda, Ratmir

Genetically encoded discovery of perfluoroaryl macrocycles that bind to albumin and exhibit extended circulation in vivo

遗传编码的全氟芳基大环化合物与白蛋白结合并在体内延长循环时间的发现

Jeffrey Y K Wong #, Arunika I Ekanayake #, Serhii Kharchenko, Steven E Kirberger, Ryan Qiu, Payam Kelich, Susmita Sarkar, Jiaqian Li, Kleinberg X Fernandez, Edgar R Alvizo-Paez, Jiayuan Miao, Shiva Kalhor-Monfared, J Dwyer John, Hongsuk Kang, Hwanho Choi, John M Nuss, John C Vederas, Yu-Shan Lin, Ma