日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

OT-82, a novel anticancer drug candidate that targets the strong dependence of hematological malignancies on NAD biosynthesis.

OT-82 是一种新型抗癌候选药物,它针对血液恶性肿瘤对 NAD 生物合成的强烈依赖性

Korotchkina Lioubov, Kazyulkin Denis, Komarov Pavel G, Polinsky Alex, Andrianova Ekaterina L, Joshi Sangeeta, Gupta Mahima, Vujcic Slavoljub, Kononov Eugene, Toshkov Ilia, Tian Yuan, Krasnov Peter, Chernov Mikhail V, Veith Jean, Antoch Marina P, Middlemiss Shiloh, Somers Klaartje, Lock Richard B, Norris Murray D, Henderson Michelle J, Haber Michelle, Chernova Olga B, Gudkov Andrei V

Central role of liver in anticancer and radioprotective activities of Toll-like receptor 5 agonist

肝脏在 Toll 样受体 5 激动剂的抗癌和放射防护活性中起着核心作用

Burdelya, Lyudmila G; Brackett, Craig M; Kojouharov, Bojidar; Gitlin, Ilya I; Leonova, Katerina I; Gleiberman, Anatoli S; Aygun-Sunar, Semra; Veith, Jean; Johnson, Christopher; Haderski, Gary J; Stanhope-Baker, Patricia; Allamaneni, Shyam; Skitzki, Joseph; Zeng, Ming; Martsen, Elena; Medvedev, Alexander; Scheblyakov, Dmitry; Artemicheva, Nataliya M; Logunov, Denis Y; Gintsburg, Alexander L; Naroditsky, Boris S; Makarov, Sergei S; Gudkov, Andrei V

Curaxins: anticancer compounds that simultaneously suppress NF-κB and activate p53 by targeting FACT

Curaxins:一种抗癌化合物,它通过靶向FACT蛋白,同时抑制NF-κB并激活p53。

Gasparian, Alexander V; Burkhart, Catherine A; Purmal, Andrei A; Brodsky, Leonid; Pal, Mahadeb; Saranadasa, Madhi; Bosykh, Dmitry A; Commane, Mairead; Guryanova, Olga A; Pal, Srabani; Safina, Alfiya; Sviridov, Sergey; Koman, Igor E; Veith, Jean; Komar, Anton A; Gudkov, Andrei V; Gurova, Katerina V