日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Comparative genomics identifies small interfering RNA with activity against all five human betacoronaviruses

比较基因组学鉴定出对所有五种人类β冠状病毒均有活性的小干扰RNA

Vogler, Julian; Ambike, Shubhankar; Velkov, Stoyan; Cheng, Cho-Chin; Neubecker, Pauline; Fischhaber, Natalie; Mallick, Pratik; Martan, Ivana; Sauerhering, Lucie; von Brunn, Albrecht; Protzer, Ulrike; Michler, Thomas

Acute testicular hyperthermia leads to rapid loss of global piRNA and a concurrent increase in LINE1 activity within heat sensitive male germ cells.

急性睾丸高温导致全身 piRNA 迅速丢失,同时热敏感雄性生殖细胞内的 LINE1 活性增加。

Robinson Benjamin R, Netherton Jacob K, Ogle Rachel A, Burnard Sean M, Williams Grace E, Tennant Georgia M, Hussein Maytham, Lee Heather J, Velkov Tony, Baker Mark A

ARRDC4-mediated glycolysis enhances innate immunity to influenza A virus through fructose-1,6-bisphosphate

ARRDC4介导的糖酵解通过果糖-1,6-二磷酸增强对甲型流感病毒的先天免疫力。

Li, Yuhan; Wang, Zhen; Wang, Jie; Jiang, Zhimin; Chen, Mingyue; Ai, Hui; Ma, Chao; Tong, Qi; Liu, Litao; Velkov, Tony; Sun, Honglei; Pu, Juan; Liu, Jinhua; Dai, Chongshan; Sun, Yipeng

Structure-Activity Relationship of the Diaminobutyric Acid Residues in Polymyxins

多粘菌素中二氨基丁酸残基的构效关系

Ma, Wendong; Jiang, Xukai; Mu, Kaijie; Tian, Sixin; Yu, Heidi H; Wickremasinghe, Hasini; Velkov, Tony; Roberts, Kade D; Patil, Nitin A; Li, Jian

SARS-CoV-2 Productively Infects Human Hepatocytes and Induces Cell Death

SARS-CoV-2 有效感染人类肝细胞并诱导细胞死亡

Chunkyu Ko, Cho-Chin Cheng, Daniele Mistretta, Shubhankar Ambike, Julia Sacherl, Stoyan Velkov, Bo-Hung Liao, Romina Bester, Merve Gültan, Olga Polezhaeva, Alexander Herrmann, Constanze A Jakwerth, Carsten B Schmidt-Weber, Joachim J Bugert, Roman Wölfel, Vincent Grass, Sandra Essbauer, Daniel Schnep

Corynoxeine Supplementation Ameliorates Colistin-Induced Kidney Oxidative Stress and Inflammation in Mice.

Corynoxeine 补充剂可改善粘菌素诱导的小鼠肾脏氧化应激和炎症

Liu Yue, Zhang Ruichen, Velkov Tony, Shen Jianzhong, Tang Shusheng, Dai Chongshan

A Comparative Review of the Pharmacology of Dalbavancin and Oritavancin for Gram-Positive Infections: Birds of a Feather or Apples and Oranges?

达巴万星和奥利万星治疗革兰氏阳性菌感染的药理学比较研究:二者是同类还是截然不同?

Hussein, Maytham; Barclay, James; Baker, Mark; Wu, Yuezhou; Thombare, Varsha J; Patil, Nitin; Murthy, Ananya B; Sharma, Rajnikant; Rao, Gauri G; Blaskovich, Mark A T; Li, Jian; Velkov, Tony

Progress of AI-Driven Drug-Target Interaction Prediction and Lead Optimization

人工智能驱动的药物靶点相互作用预测和先导化合物优化进展

Wang, Qiqi; Sun, Boyan; Yi, Yunpeng; Velkov, Tony; Shen, Jianzhong; Dai, Chongshan; Jiang, Haiyang

Hyperforin potentiates polymyxin B against multidrug-resistant Gram-negative pathogens via membrane disruption, biofilm eradication, and oxidative stress

金丝桃素通过破坏细胞膜、清除生物膜和氧化应激增强多粘菌素B对抗多重耐药革兰氏阴性病原体的疗效。

Hussein, Maytham; Crawford, Simon; Baker, Mark; Floyd, Holly; Allobawi, Rafah; Blaskovich, Mark A T; Rao, Gauri G; Zuegg, Johannes; Li, Jian; Velkov, Tony

Prolonged exposure to teixobactin generates cross-tolerance to other cell wall-targeting antimicrobials in Enterococcus faecalis

长期接触替索巴汀会导致粪肠球菌对其他靶向细胞壁的抗菌药物产生交叉耐受性。

Darnell, Rachel L; Knottenbelt, Melanie K; Rose, Olivia E; Cleary, Caitlin S B; Todd Rose, Francesca O; Hodgkinson, Hannah; Wu, Yuezhou; Hussein, Maytham; Velkov, Tony; Gebhard, Susanne; Cook, Gregory M