日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Activity Relationship of Antischistosomal Aryl Hydantoin (AR102)

抗血吸虫药芳基乙内酰脲(AR102)的构效关系

Leas, Derek A; Häberli, Cécile; White, Karen L; Shackleford, David M; Jones, Jeremy O; Campbell, Michael; Wu, Jianbo; Kaushik, Deepender; Dong, Yuxiang; Wallick, Alexander I; Charman, Susan A; Keiser, Jennifer; Davis, Paul H; Vennerstrom, Jonathan L

Spleen and peripheral blood immunopathology in an outbred model of adult-stage murine schistosomiasis

成年小鼠血吸虫病近交系模型中脾脏和外周血的免疫病理学

Schulze, Thomas T; Neville, Andrew J; Ehrhorn, Evie G; Alsuleiman, Sarah A; Vennerstrom, Jonathan L; Davis, Paul H

Comparative Hydrophobicity, Solubility, and Metabolic Stability of 4(1H)-Pyridones, 4(1H)-Quinolones, and 9(10H)-Acridones

4(1H)-吡啶酮、4(1H)-喹诺酮和9(10H)-吖啶酮的疏水性、溶解度和代谢稳定性比较

Ren, Rongguo; Zhong, Longjin; Noack, Cassandra; Kaushik, Deepender; Leas, Derek A; Wang, Xiaofang; Dong, Yuxiang; Charman, Susan A; Vennerstrom, Jonathan L

Single-Dose Drug Development Candidate for Schistosomiasis

血吸虫病单剂量药物研发候选药物

Leas, Derek A; Keiser, Jennifer; Charman, Susan A; Shackleford, David M; Jones, Jeremy O; Campbell, Michael; Chen, Gong; Katneni, Kasiram; Patil, Rahul; Hu, Meiyu; Pham, Thao; Häberli, Cécile; Schulze, Thomas T; Neville, Andrew J; Wang, Xiaofang; Dong, Yuxiang; Davis, Paul H; Vennerstrom, Jonathan L

Antimalarial Dibenzannulated Medium-Ring Keto Lactams

抗疟疾二苯并环中环酮内酰胺类药物

Ren, Rongguo; Wang, Xiaofang; Leas, Derek A; Scheurer, Christian; Hoevel, Sarah; Cal, Monica; Chen, Gong; Zhong, Longjin; Katneni, Kasiram; Pham, Thao; Patil, Rahul; Sil, Diptesh; Walters, Matthias J; Schulze, Thomas T; Neville, Andrew J; Dong, Yuxiang; Wittlin, Sergio; Kaiser, Marcel; Davis, Paul H; Charman, Susan A; Vennerstrom, Jonathan L

Synthesis and antimalarial activity of amide and ester conjugates of siderophores and ozonides

铁载体和臭氧化物酰胺和酯缀合物的合成及其抗疟活性

Tiwari, Rohit; Checkley, Lisa; Ferdig, Michael T; Vennerstrom, Jonathan L; Miller, Marvin J

Metabolic, Pharmacokinetic, and Activity Profile of the Liver Stage Antimalarial (RC-12)

肝期抗疟药(RC-12)的代谢、药代动力学和活性特征

Dong, Yuxiang; Sonawane, Yogesh; Maher, Steven P; Zeeman, Anne-Marie; Chaumeau, Victor; Vantaux, Amélie; Cooper, Caitlin A; Chiu, Francis C K; Ryan, Eileen; McLaren, Jenna; Chen, Gong; Wittlin, Sergio; Witkowski, Benoît; Nosten, François; Sriraghavan, Kamaraj; Kyle, Dennis E; Kocken, Clemens H M; Charman, Susan A; Vennerstrom, Jonathan L

Peroxide Antimalarial Drugs Target Redox Homeostasis in Plasmodium falciparum Infected Red Blood Cells

过氧化物抗疟药靶向恶性疟原虫感染红细胞中的氧化还原稳态

Ghizal Siddiqui, Carlo Giannangelo, Amanda De Paoli, Anna Katharina Schuh, Kim C Heimsch, Dovile Anderson, Timothy G Brown, Christopher A MacRaild, Jianbo Wu, Xiaofang Wang, Yuxiang Dong, Jonathan L Vennerstrom, Katja Becker, Darren J Creek

Antischistosomal tetrahydro-γ-carboline sulfonamides

抗血吸虫四氢-γ-咔啉磺酰胺

Ren, Rongguo; Wang, Xiaofang; Leas, Derek A; Häberli, Cécile; Cal, Monica; Dong, Yuxiang; Kaiser, Marcel; Keiser, Jennifer; Vennerstrom, Jonathan L

In Vitro Selection Implicates ROP1 as a Resistance Gene for an Experimental Therapeutic Benzoquinone Acyl Hydrazone in Toxoplasma gondii

体外筛选表明 ROP1 是弓形虫中一种实验性治疗用苯醌酰腙的抗性基因

Martens, Matthew C; Won, Madalyn M; Won, Harim I; Schulze, Thomas T; Judge, Abigail K; Neville, Andrew J; Vennerstrom, Jonathan L; Davis, Paul H