日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A µ-opioid receptor superagonist analgesic with minimal adverse effects

一种μ-阿片受体超激动剂镇痛药,不良反应极小

Gomez, Juan L; Ventriglia, Emilya N; Frangos, Zachary J; Sulima, Agnieszka; Robertson, Michael J; Sacco, Michael D; Budinich, Reece C; Giosan, Ilinca M; Xie, Tongzhen; Solis, Oscar; Tischer, Anna E; Bossert, Jennifer M; Caldwell, Kiera E; Bonbrest, Hannah; Essmann, Amelie; Garçon-Poca, Zelai M; Choi, Shinbe; Noya, Michael R; Limiac, Feonil; Arce, Ali; Glatfelter, Grant C; Robinson, Margaret; Chen, Li; Mullarkey, Angelina A; Brademan, Dain R; Enten, Garrett; Dunne, William; Quiroz, César; Schoenborn, Ingrid; Lee, Chae Bin; Rais, Rana; Holt, Daniel P; Dannals, Robert F; Shi, Lei; Hüttenhain, Ruth; Ferré, Sergi; Kiyatkin, Eugene; Bonaventura, Jordi; Shaham, Yavin; Zachariou, Venetia; Baumann, Michael H; Skiniotis, Georgios; Rice, Kenner C; Michaelides, Michael

An emerging role for synaptic Zn(2+) in substance use disorders

突触锌离子(Zn(2+))在物质使用障碍中的新兴作用

Solis, Oscar; Curry, Fallon P; Frangos, Zachary J; Dunne, William; Schoenborn, Ingrid; Lauer, Alyssa; Gomez, Juan L; Ventriglia, Emilya N; Bonaventura, Jordi; Michaelides, Michael

D2 autoreceptors gate vulnerability to cocaine use disorder

D2自身受体控制对可卡因使用障碍的易感性

Murray, Erin M; Diaz-Urbina, Daniel; Bock, Roland; Ventriglia, Emilya; Tischer, Anna; Shin, Jung Hoon; Lee, Seul Ah; Anderson, Lucy G; Cerveny, Sydney; Bleimeister, Isabel; Bocarsly, Miriam E; Michaelides, Michael; Alvarez, Veronica A

Cocaine chemogenetics blunts drug-seeking by synthetic physiology.

可卡因化学遗传学通过合成生理学抑制药物渴求。

Gomez Juan L, Magnus Christopher J, Bonaventura Jordi, Solis Oscar, Curry Fallon P, Levinstein Marjorie R, Budinich Reece C, Carlton Meghan L, Ventriglia Emilya N, Lam Sherry, Wang Le, Schoenborn Ingrid, Dunne William, Michaelides Michael, Sternson Scott M

Preexisting risk-avoidance and enhanced alcohol relief are driven by imbalance of the striatal dopamine receptors in mice

小鼠纹状体多巴胺受体失衡驱动了其既有的风险规避行为和增强的酒精缓解作用。

Bocarsly, Miriam E; Shaw, Marlisa J; Ventriglia, Emilya; Anderson, Lucy G; Goldbach, Hannah C; Teresi, Catherine E; Bravo, Marilyn; Bock, Roland; Hong, Patrick; Kwon, Han Bin; Khawaja, Imran M; Raman, Rishi; Murray, Erin M; Bonaventura, Jordi; Burke, Dennis A; Michaelides, Michael; Alvarez, Veronica A

Unique pharmacodynamic properties and low abuse liability of the µ-opioid receptor ligand (S)-methadone

μ-阿片受体配体(S)-美沙酮具有独特的药效学特性和低滥用风险

Levinstein, Marjorie R; De Oliveira, Paulo A; Casajuana-Martin, Nil; Quiroz, Cesar; Budinich, Reece C; Rais, Rana; Rea, William; Ventriglia, Emilya N; Llopart, Natàlia; Casadó-Anguera, Verònica; Moreno, Estefanía; Walther, Donna; Glatfelter, Grant C; Weinshenker, David; Zarate, Carlos A Jr; Casadó, Vicent; Baumann, Michael H; Pardo, Leonardo; Ferré, Sergi; Michaelides, Michael

In vivo photopharmacology with light-activated opioid drugs.

利用光激活阿片类药物进行体内光药理学研究

McClain Shannan P, Ma Xiang, Johnson Desiree A, Johnson Caroline A, Layden Aryanna E, Yung Jean C, Lubejko Susan T, Livrizzi Giulia, He X Jenny, Zhou Jingjing, Chang-Weinberg Janie, Ventriglia Emilya, Rizzo Arianna, Levinstein Marjorie, Gomez Juan L, Bonaventura Jordi, Michaelides Michael, Banghart Matthew R

Mu Opioid Receptor Activation Mediates (S)-ketamine Reinforcement in Rats: Implications for Abuse Liability

μ阿片受体激活介导(S)-氯胺酮在大鼠体内的强化作用:对滥用责任的启示

Levinstein, Marjorie R; Carlton, Meghan L; Di Ianni, Tommaso; Ventriglia, Emilya N; Rizzo, Arianna; Gomez, Juan L; Budinich, Reece C; Shaham, Yavin; Airan, Raag D; Zarate, Carlos A Jr; Bonaventura, Jordi; Michaelides, Michael

Essential role of P-glycoprotein in the mechanism of action of oliceridine

P-糖蛋白在奥利西啶作用机制中的关键作用

Ventriglia, Emilya; Rizzo, Arianna; Gomez, Juan L; Friedman, Jacob; Lam, Sherry; Solís, Oscar; Rais, Rana; Bonaventura, Jordi; Michaelides, Michael

6-O-(2-[(18)F]Fluoroethyl)-6-O-Desmethyl-Diprenorphine ([(18)F]FE-DPN) Preferentially Binds to Mu Opioid Receptors In Vivo

6-O-(2-[(18)F]氟乙基)-6-O-去甲基-二丙诺啡 ([(18)F]FE-DPN) 在体内优先与μ阿片受体结合

Levinstein, Marjorie R; Ventriglia, Emilya N; Gomez, Juan L; Budinich, Reece C; Marton, János; Henriksen, Gjermund; Holt, Daniel P; Dannals, Robert F; Pomper, Martin G; Zarate, Carlos A Jr; Bonaventura, Jordi; Michaelides, Michael