日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Enhanced anticancer effect of thymidylate synthase dimer disrupters by promoting intracellular accumulation.

胸苷酸合成酶二聚体破坏剂通过促进细胞内积累增强抗癌作用

Marverti Gaetano, Moschella Maria Gaetana, Belardo Alice, Lamesta Michele, Mercanile Giada, Tagliazucchi Lorenzo, Aiello Daniele, Venturelli Alberto, Illuminati Davide, Guerrini Remo, Losi Lorena, Ponterini Glauco, Costi Maria Paola, D'Arca Domenico

Antitarget, Anti-SARS-CoV-2 Leads, Drugs, and the Drug Discovery-Genetics Alliance Perspective

抗靶点、抗SARS-CoV-2先导化合物、药物以及药物发现-遗传学联盟的展望

Pozzi, Cecilia; Vanet, Anne; Francesconi, Valeria; Tagliazucchi, Lorenzo; Tassone, Giusy; Venturelli, Alberto; Spyrakis, Francesca; Mazzorana, Marco; Costi, Maria P; Tonelli, Michele

Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1

多靶点选择性化合物设计获得了强效的动质体蝶呤还原酶抑制剂 1

Pöhner, Ina; Quotadamo, Antonio; Panecka-Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Costi, Maria P; Venturelli, Alberto; Wade, Rebecca C

Current Treatments to Control African Trypanosomiasis and One Health Perspective

目前控制非洲锥虫病的治疗方法及一体化健康视角

Venturelli, Alberto; Tagliazucchi, Lorenzo; Lima, Clara; Venuti, Federica; Malpezzi, Giulia; Magoulas, George E; Santarem, Nuno; Calogeropoulou, Theodora; Cordeiro-da-Silva, Anabela; Costi, Maria Paola

Virtual screening identifies broad-spectrum β-lactamase inhibitors with activity on clinically relevant serine- and metallo-carbapenemases

虚拟筛选可鉴定出对临床相关的丝氨酸和金属碳青霉烯酶具有活性的广谱β-内酰胺酶抑制剂。

Spyrakis, Francesca; Santucci, Matteo; Maso, Lorenzo; Cross, Simon; Gianquinto, Eleonora; Sannio, Filomena; Verdirosa, Federica; De Luca, Filomena; Docquier, Jean-Denis; Cendron, Laura; Tondi, Donatella; Venturelli, Alberto; Cruciani, Gabriele; Costi, Maria Paola