Deuterated buprenorphine retains pharmacodynamic properties of buprenorphine and resists metabolism to the active metabolite norbuprenorphine in rats
氘代丁丙诺啡保留了丁丙诺啡的药效学特性,并且抵抗大鼠体内活性代谢物去甲丁丙诺啡的代谢
期刊:Frontiers in Pharmacology
影响因子:4.4
doi:10.3389/fphar.2023.1123261
Venumadhav Janganati, Paloma Salazar, Brian J Parks, Gregory S Gorman, Paul L Prather, Eric C Peterson, Alexander W Alund, Jeffery H Moran, Peter A Crooks, Lisa K Brents