UK-78,282, a novel piperidine compound that potently blocks the Kv1.3 voltage-gated potassium channel and inhibits human T cell activation
UK-78,282 是一种新型哌啶化合物,能有效阻断 Kv1.3 电压门控钾通道并抑制人 T 细胞活化。
期刊:British Journal of Pharmacology
影响因子:7.7
doi:10.1038/sj.bjp.0702480
Hanson, D C; Nguyen, A; Mather, R J; Rauer, H; Koch, K; Burgess, L E; Rizzi, J P; Donovan, C B; Bruns, M J; Canniff, P C; Cunningham, A C; Verdries, K A; Mena, E; Kath, J C; Gutman, G A; Cahalan, M D; Grissmer, S; Chandy, K G