日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Design, Synthesis, and Biological Evaluation of the Cage-Amide Derived Orthopox Virus Replication Inhibitors

基于结构的笼酰胺衍生正痘病毒复制抑制剂的设计、合成和生物学评价

Evgenii S Mozhaitsev ,Evgeniy V Suslov ,Daria A Rastrepaeva ,Olga I Yarovaya ,Sophia S Borisevich ,Edward M Khamitov ,Dmitry S Kolybalov ,Sergey G Arkhipov ,Nikolai I Bormotov ,Larisa N Shishkina ,Olga A Serova ,Roman V Brunilin ,Andrey A Vernigora ,Maxim B Nawrozkij ,Alexander P Agafonov ,Rinat A Maksyutov ,Konstantin P Volcho ,Nariman F Salakhutdinov

Ureas derived from camphor and fenchone reveal enantiomeric preference of human soluble epoxide hydrolase

樟脑和芬酮衍生的脲类化合物揭示了人可溶性环氧化物水解酶的对映体偏好性

Vladimir Burmistrov ,Christophe Morisseau ,Dmitry Pitushkin ,Robert R Fayzullin ,Dmitry Karlov ,Andrey Vernigora ,Yaroslav Kuznetsov ,Saeef M H Abbas ,Gennady M Butov ,Bruce D Hammock

Bioisosteric substitution of adamantane with bicyclic lipophilic groups improves water solubility of human soluble epoxide hydrolase inhibitors

金刚烷与双环亲脂基团的生物等排取代可提高人可溶性环氧化物水解酶抑制剂的水溶性。

Burmistrov, Vladimir; Morisseau, Christophe; Karlov, Dmitry; Pitushkin, Dmitry; Vernigora, Andrey; Rasskazova, Elena; Butov, Gennady M; Hammock, Bruce D