日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of a Highly Cooperative PROTAC Degrader Targeting GTP-Loaded KRAS(On) Alleles

鉴定一种高度协同的PROTAC降解酶,该酶靶向GTP结合的KRAS(On)等位基因

Vetma, Vesna; Puoti, Ilaria; Karolak, Natalia K; Chakraborti, Sohini; Diers, Emelyne; Girardi, Enrico; Khan, Shakil; Kidd, Giorgia; Kropatsch, Katrin G; Mclennan, Ross; O'Connor, Suzanne; Samwer, Matthias; Trainor, Nicole; Whitworth, Claire; Wijaya, Andre J; Wong, Jeff Y F; Zollman, David; Farnaby, William; Popow, Johannes; Ciulli, Alessio; Ettmayer, Peter; McAulay, Kirsten

Use of Aldehyde-Alkyne-Amine Couplings to Generate Medicinal Chemistry-Relevant Linkers

利用醛-炔-胺偶联反应生成与药物化学相关的连接基

McGown, Andrew; Vetma, Vesna; Crepin, Damien; Lin, Yan; Adcock, Claire; Craigon, Conner; Nafie, Jordan; von Emloh, Daniel; Sutton, Léa; Bailey, Kiera; Edmunds, Lewis; Sharma, Manvendra; Wilden, Jonathan D; Coles, Simon J; Tizzard, Graham J; Farnaby, William; Ciulli, Alessio; Kostakis, George E; Spencer, John

Tuning the open-close equilibrium of Cereblon with small molecules influences protein degradation

利用小分子调节 Cereblon 的开闭平衡会影响蛋白质降解

O'Connor, Suzanne; Rutter, Zoe J; Cowan, Angus D; Zeeb, Markus; Binder, Florian; Cao, Yuting; Chakraborti, Sohini; Djukic, Stefan; Geist, Leonhard; Hogg, Elizabeth; Kidd, Giorgia; Krumb, Matthias; Langer, Simon; Schmidt, Denis; Martin, Liam; McCrory, Elisha H; Padroni, Giacomo; Puoti, Ilaria; Simpson, Luke; Sturbaut, Manon; Crozier, Lisa; Vetma, Vesna; Zhang, Qingzhi; McAulay, Kirsten; Theis, Theodor; Ciulli, Alessio

Convergence of pathway analysis and pattern recognition predicts sensitization to latest generation TRAIL therapeutics by IAP antagonism.

通路分析和模式识别的融合预测了IAP拮抗作用对最新一代TRAIL疗法的敏感性

Vetma Vesna, Guttà Cristiano, Peters Nathalie, Praetorius Christian, Hutt Meike, Seifert Oliver, Meier Friedegund, Kontermann Roland, Kulms Dagmar, Rehm Markus

Optimization of an ex vivo gene transfer to the hamstrings tendons muscle remnants: potential for genetic enhancement of bone healing

优化体外基因转移至腘绳肌腱残余组织:增强骨愈合的基因潜力

Rod, Eduard; Matić, Igor; Antunović, Maja; Vetma, Vesna; Pavičić, Ivan; Hudetz, Damir; Marijanović, Inga; Primorac, Dragan; Ivković, Alan

Examining the In Vitro Efficacy of the IAP Antagonist Birinapant as a Single Agent or in Combination With Dacarbazine to Induce Melanoma Cell Death

体外研究IAP拮抗剂Birinapant作为单药或与达卡巴嗪联合用药诱导黑色素瘤细胞死亡的功效

Vetma, Vesna; Rožanc, Jan; Charles, Emilie M; Hellwig, Christian T; Alexopoulos, Leonidas G; Rehm, Markus