日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dual targeting of the androgen receptor and PI3K/AKT/mTOR pathways in prostate cancer models improves antitumor efficacy and promotes cell apoptosis

在前列腺癌模型中,雄激素受体和 PI3K/AKT/mTOR 通路的双重靶向可提高抗肿瘤功效并促进细胞凋亡

Tatsuo Sugawara, Ekaterina Nevedomskaya, Simon Heller, Annika Böhme, Ralf Lesche, Oliver von Ahsen, Sylvia Grünewald, Holly M Nguyen, Eva Corey, Simon J Baumgart, Victoria Georgi, Vera Pütter, Amaury Fernández-Montalván, James D Vasta, Matthew B Robers, Oliver Politz, Dominik Mumberg, Bernard Haendl

A miniaturized mode-of-action profiling platform enables high throughput characterization of the molecular and cellular dynamics of EZH2 inhibition

微型作用模式分析平台能够高通量表征 EZH2 抑制的分子和细胞动力学

Lilia Falkenstern #, Victoria Georgi #, Stefanie Bunse, Volker Badock, Manfred Husemann, Ulrike Roehn, Timo Stellfeld, Mark Fitzgerald, Steven Ferrara, Detlef Stöckigt, Carlo Stresemann, Ingo V Hartung, Amaury Fernández-Montalván

In vitro and in silico analysis of the effects of D2 receptor antagonist target binding kinetics on the cellular response to fluctuating dopamine concentrations

体外和计算机模拟分析 D2 受体拮抗剂靶标结合动力学对细胞对波动的多巴胺浓度反应的影响

Wilhelmus E A de Witte, Joost W Versfelt, Maria Kuzikov, Solene Rolland, Victoria Georgi, Philip Gribbon, Sheraz Gul, Dymphy Huntjens, Piet Hein van der Graaf, Meindert Danhof, Amaury Fernández-Montalván, Gesa Witt, Elizabeth C M de Lange