A Divergent SAR Study Allows Optimization of a Potent 5-HT2c Inhibitor to a Promising Antimalarial Scaffold
一项不同的构效关系研究使得一种强效的5-HT2c抑制剂能够优化为一种有前景的抗疟疾骨架。
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/ml300008j
Calderón, Félix; Vidal-Mas, Jaume; Burrows, Jeremy; de la Rosa, Juan Carlos; Jiménez-Díaz, María Belén; Mulet, Teresa; Prats, Sara; Solana, Jorge; Witty, Michael; Gamo, Francisco Javier; Fernández, Esther