A selective BCL-XL PROTAC degrader achieves safe and potent antitumor activity
一种选择性BCL-XL PROTAC降解剂可实现安全有效的抗肿瘤活性
期刊:Nature Medicine
影响因子:58.7
doi:10.1038/s41591-019-0668-z
Sajid Khan # ,Xuan Zhang # ,Dongwen Lv # ,Qi Zhang ,Yonghan He ,Peiyi Zhang ,Xingui Liu ,Dinesh Thummuri ,Yaxia Yuan ,Janet S Wiegand ,Jing Pei ,Weizhou Zhang ,Abhisheak Sharma ,Christopher R McCurdy ,Vinitha M Kuruvilla ,Natalia Baran ,Adolfo A Ferrando ,Yong-Mi Kim ,Anna Rogojina ,Peter J Houghton ,Guangcun Huang ,Robert Hromas ,Marina Konopleva ,Guangrong Zheng ,Daohong Zhou