日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Hypoxia-Activated Prodrug TH-302 Targets Hypoxic Bone Marrow Niches in Preclinical Leukemia Models

缺氧激活前药TH-302靶向临床前白血病模型中的缺氧骨髓微环境

Benito, Juliana; Ramirez, Marc S; Millward, Niki Zacharias; Velez, Juliana; Harutyunyan, Karine G; Lu, Hongbo; Shi, Yue-Xi; Matre, Polina; Jacamo, Rodrigo; Ma, Helen; Konoplev, Sergej; McQueen, Teresa; Volgin, Andrei; Protopopova, Marina; Mu, Hong; Lee, Jaehyuk; Bhattacharya, Pratip K; Marszalek, Joseph R; Davis, R Eric; Bankson, James A; Cortes, Jorge E; Hart, Charles P; Andreeff, Michael; Konopleva, Marina

Synthesis and preliminary evaluation of [18F]-labeled 2-oxoquinoline derivatives for PET imaging of cannabinoid CB2 receptor

合成并初步评价[18F]标记的2-氧代喹啉衍生物用于大麻素CB2受体的PET成像

Turkman, Nashaat; Shavrin, Aleksander; Paolillo, Vincenzo; Yeh, Hsin Hsien; Flores, Leo; Soghomonian, Suren; Rabinovich, Brian; Volgin, Andrei; Gelovani, Juri; Alauddin, Mian

HIF-1-dependent stromal adaptation to ischemia mediates in vivo tumor radiation resistance.

HIF-1依赖的基质对缺血的适应介导体内肿瘤放射抗性

Schwartz David L, Bankson James, Bidaut Luc, He Yi, Williams Ryan, Lemos Robert, Thitai Arun Kumar, Oh Junghwan, Volgin Andrei, Soghomonyan Suren, Yeh Hsin-Hsien, Nishii Ryuichi, Mukhopadhay Uday, Alauddin Mian, Mushkudiani Ioseb, Kuno Norihito, Krishnan Sunil, Bornman William, Lai Stephen Y, Powis Garth, Hazle John, Gelovani Juri

Fluorinated cannabinoid CB2 receptor ligands: synthesis and in vitro binding characteristics of 2-oxoquinoline derivatives.

氟化大麻素 CB2 受体配体:2-氧代喹啉衍生物的合成及体外结合特性

Turkman Nashaat, Shavrin Aleksander, Ivanov Roman A, Rabinovich Brian, Volgin Andrei, Gelovani Juri G, Alauddin Mian M

Radiosynthesis and initial in vitro evaluation of [18F]F-PEG6-IPQA--a novel PET radiotracer for imaging EGFR expression-activity in lung carcinomas

[18F]F-PEG6-IPQA 的放射合成及初步体外评价——一种用于肺癌中 EGFR 表达活性成像的新型 PET 放射性示踪剂

Pal, Ashutosh; Balatoni, Julius A; Mukhopadhyay, Uday; Ogawa, Kazuma; Gonzalez-Lepera, Carlos; Shavrin, Aleksandr; Volgin, Andrei; Tong, William; Alauddin, Mian M; Gelovani, Juri G

The selective hypoxia inducible factor-1 inhibitor PX-478 provides in vivo radiosensitization through tumor stromal effects

选择性缺氧诱导因子-1抑制剂PX-478通过肿瘤基质效应提供体内放射增敏作用。

Schwartz, David L; Powis, Garth; Thitai-Kumar, Arun; He, Yi; Bankson, James; Williams, Ryan; Lemos, Robert; Oh, Junghwan; Volgin, Andrei; Soghomonyan, Suren; Nishii, Ryuichi; Alauddin, Mian; Mukhopadhay, Uday; Peng, Zhenghong; Bornmann, William; Gelovani, Juri

Detection of pancreatic carcinomas by imaging lactose-binding protein expression in peritumoral pancreas using [18F]fluoroethyl-deoxylactose PET/CT

利用[18F]氟乙基脱氧乳糖PET/CT成像技术检测肿瘤周围胰腺中乳糖结合蛋白的表达,从而诊断胰腺癌

Flores, Leo Garcia; Bertolini, Susanna; Yeh, Hsin Hsin; Young, Daniel; Mukhopadhyay, Uday; Pal, Ashutosh; Ying, Yunming; Volgin, Andrei; Shavrin, Aleksandr; Soghomonyan, Suren; Tong, William; Bornmann, William; Alauddin, Mian M; Logsdon, Craig; Gelovani, Juri G